Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 765
LigandChemical structure of BindingDB Monomer ID 5828BDBM5828(1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-{4-[methy...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
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Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5829BDBM5829(1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-{4-[methy...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5827BDBM5827(1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-{4-[(2-{[...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5832BDBM5832(3-{4-[methyl({2-[(3-sulfamoylphenyl)amino]pyrimidi...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5833BDBM5833(3-{4-[methyl({2-[(4-sulfamoylphenyl)amino]pyrimidi...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
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Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5830BDBM5830(1-(4-acetylphenyl)-3-{4-[(2-{[3-(methanesulfonylme...)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5844BDBM5844(3-{4-[(2-{[4-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5831BDBM5831(3-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5835BDBM5835(3-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
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Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5836BDBM5836(3-ethyl-1-{4-[(2-{[3-(methanesulfonylmethyl)phenyl...)
Affinity DataIC50: 17nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5837BDBM5837(3-ethyl-1-{4-[(2-{[4-(methanesulfonylmethyl)phenyl...)
Affinity DataIC50: 26nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5838BDBM5838(3-butyl-1-{4-[(2-{[3-(methanesulfonylmethyl)phenyl...)
Affinity DataIC50: 29nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
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Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5839BDBM5839(3-cyclopentyl-1-{4-[(2-{[3-(methanesulfonylmethyl)...)
Affinity DataIC50: 31nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5826BDBM5826(1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-{4-[(2-{[...)
Affinity DataIC50: 35nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5834BDBM5834(1-(2,6-dichlorophenyl)-3-{4-[(2-{[3-(methanesulfon...)
Affinity DataIC50: 65nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5845BDBM5845(3-{4-[(2-{[4-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5840BDBM5840(3-[2-(dimethylamino)ethyl]-1-{4-[(2-{[3-(methanesu...)
Affinity DataIC50: 681nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5842BDBM5842(3-{4-[(2-{[4-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 990nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5841BDBM5841(3-[2-(dimethylamino)ethyl]-1-{4-[(2-{[4-(methanesu...)
Affinity DataIC50: 3.11E+3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5843BDBM5843(N-{4-[(2-{[4-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 4.49E+3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed