Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50016495
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20330BDBM20330(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataKi:  3.40nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20321BDBM20321(JYL1421 | CHEMBL388824 | 3-[(4-tert-butylphenyl)me...)
Affinity DataKi:  9.16nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20330BDBM20330(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataKi:  50.4nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20321BDBM20321(JYL1421 | CHEMBL388824 | 3-[(4-tert-butylphenyl)me...)
Affinity DataKi:  53.5nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20315BDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataKi:  54nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20315BDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataKi:  63nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169732BDBM50169732((4-tert-Butyl-benzyl)-thiocarbamic acid 4-methanes...)
Affinity DataKi:  110nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169728BDBM50169728(N-(4-tert-Butyl-benzyl)-2-(3-fluoro-4-methanesulfo...)
Affinity DataKi:  118nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169733BDBM50169733((4-tert-Butyl-benzyl)-thiocarbamic acid 3-fluoro-4...)
Affinity DataKi:  120nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169735BDBM50169735((4-tert-Butyl-benzyl)-thiocarbamic acid 4-methanes...)
Affinity DataKi:  222nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169740BDBM50169740(N-{4-[3-(4-tert-Butyl-benzyl)-ureidomethyl]-phenyl...)
Affinity DataKi:  225nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169726BDBM50169726(N-(4-tert-Butyl-benzyl)-2-(4-methanesulfonylamino-...)
Affinity DataKi:  398nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169733BDBM50169733((4-tert-Butyl-benzyl)-thiocarbamic acid 3-fluoro-4...)
Affinity DataKi:  450nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169732BDBM50169732((4-tert-Butyl-benzyl)-thiocarbamic acid 4-methanes...)
Affinity DataKi:  461nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169734BDBM50169734(N-{(4-tert-butylbenzyl)-N'-hydroxythiourea}methyl)...)
Affinity DataKi:  470nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169722BDBM50169722(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)p...)
Affinity DataKi:  470nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169728BDBM50169728(N-(4-tert-Butyl-benzyl)-2-(3-fluoro-4-methanesulfo...)
Affinity DataKi:  472nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20284BDBM20284(N-[2-(4-chlorophenyl)ethyl]-7,8-dihydroxy-2,3,4,5-...)
Affinity DataKi:  520nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169717BDBM50169717(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)2...)
Affinity DataKi:  579nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169738BDBM50169738(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)2...)
Affinity DataKi:  635nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169735BDBM50169735((4-tert-Butyl-benzyl)-thiocarbamic acid 4-methanes...)
Affinity DataKi:  772nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169727BDBM50169727(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)2...)
Affinity DataKi:  800nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169724BDBM50169724(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)2...)
Affinity DataKi:  926nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169722BDBM50169722(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)p...)
Affinity DataKi:  1.09E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20284BDBM20284(N-[2-(4-chlorophenyl)ethyl]-7,8-dihydroxy-2,3,4,5-...)
Affinity DataKi:  1.30E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169717BDBM50169717(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)2...)
Affinity DataKi:  1.31E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169738BDBM50169738(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)2...)
Affinity DataKi:  1.33E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169719BDBM50169719(N-(4-tert-butylbenzyl)-2-{4-[(methylsulfonyl)amino...)
Affinity DataKi:  1.46E+3nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169730BDBM50169730(N-{4-[(methylsulfonyl)amino]benzyl}2-(4-tert-butyl...)
Affinity DataKi:  2.01E+3nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169726BDBM50169726(N-(4-tert-Butyl-benzyl)-2-(4-methanesulfonylamino-...)
Affinity DataKi:  2.10E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169718BDBM50169718((4-Methanesulfonylamino-3-methoxy-benzyl)-thiocarb...)
Affinity DataKi:  2.17E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169721BDBM50169721(N-{(4-tert-butylbenzyl)-N-hydroxythiourea}methyl)3...)
Affinity DataKi:  2.27E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169740BDBM50169740(N-{4-[3-(4-tert-Butyl-benzyl)-ureidomethyl]-phenyl...)
Affinity DataKi:  2.56E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169731BDBM50169731(N-[3-(3,4-Dimethyl-phenyl)-propyl]-2-(3-fluoro-4-m...)
Affinity DataKi:  2.71E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169723BDBM50169723(N-{(4-tert-butylbenzyl)-N'-hydroxyurea}methyl)phen...)
Affinity DataKi:  3.50E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169734BDBM50169734(N-{(4-tert-butylbenzyl)-N'-hydroxythiourea}methyl)...)
Affinity DataKi:  4.26E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169737BDBM50169737((4-Methanesulfonylamino-benzyl)-thiocarbamic acid ...)
Affinity DataKi:  4.60E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169731BDBM50169731(N-[3-(3,4-Dimethyl-phenyl)-propyl]-2-(3-fluoro-4-m...)
Affinity DataKi:  4.66E+3nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169725BDBM50169725(2-(4-tert-Butyl-phenyl)-N-(4-methanesulfonylamino-...)
Affinity DataKi:  5.22E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169736BDBM50169736(2-(4-tert-Butyl-phenyl)-N-hydroxy-N-(4-methanesulf...)
Affinity DataKi:  5.30E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169737BDBM50169737((4-Methanesulfonylamino-benzyl)-thiocarbamic acid ...)
Affinity DataKi:  6.25E+3nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169720BDBM50169720(N-(4-tert-Butyl-benzyl)-N-hydroxy-2-(4-methanesulf...)
Affinity DataKi:  6.40E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169730BDBM50169730(N-{4-[(methylsulfonyl)amino]benzyl}2-(4-tert-butyl...)
Affinity DataKi:  6.40E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169720BDBM50169720(N-(4-tert-Butyl-benzyl)-N-hydroxy-2-(4-methanesulf...)
Affinity DataKi:  6.60E+3nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169725BDBM50169725(2-(4-tert-Butyl-phenyl)-N-(4-methanesulfonylamino-...)
Affinity DataKi:  6.76E+3nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169729BDBM50169729(N-[3-(3,4-Dimethyl-phenyl)-propyl]-2-(4-methanesul...)
Affinity DataKi:  7.18E+3nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169718BDBM50169718((4-Methanesulfonylamino-3-methoxy-benzyl)-thiocarb...)
Affinity DataKi:  8.40E+3nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169719BDBM50169719(N-(4-tert-butylbenzyl)-2-{4-[(methylsulfonyl)amino...)
Affinity DataKi:  1.21E+4nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169729BDBM50169729(N-[3-(3,4-Dimethyl-phenyl)-propyl]-2-(4-methanesul...)
Affinity DataKi:  1.36E+4nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169739BDBM50169739(2-(4-Methanesulfonylamino-phenyl)-N-octadec-9-enyl...)
Affinity DataKi: >2.50E+4nMAssay Description:In vitro inhibition of [3H]RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed