Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50041382
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410041BDBM50410041(CHEMBL178951)
Affinity DataKi:  0.0182nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410036BDBM50410036(CHEMBL179761)
Affinity DataKi:  0.0871nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410038BDBM50410038(CHEMBL179103)
Affinity DataKi:  0.251nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410028BDBM50410028(CHEMBL359753)
Affinity DataKi:  0.302nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410031BDBM50410031(CHEMBL362069)
Affinity DataKi:  0.490nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410042BDBM50410042(CHEMBL366431)
Affinity DataKi:  1.41nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410032BDBM50410032(CHEMBL361980)
Affinity DataKi:  1.51nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410045BDBM50410045(CHEMBL179250)
Affinity DataKi:  1.70nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410027BDBM50410027(CHEMBL180816)
Affinity DataKi:  2.51nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410034BDBM50410034(CHEMBL181166)
Affinity DataKi:  4.90nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410035BDBM50410035(CHEMBL181514)
Affinity DataKi:  7.94nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410039BDBM50410039(CHEMBL179367)
Affinity DataKi:  11.0nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410037BDBM50410037(CHEMBL178277)
Affinity DataKi:  15.1nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410044BDBM50410044(CHEMBL361999)
Affinity DataKi:  550nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410043BDBM50410043(CHEMBL180655)
Affinity DataKi:  776nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410033BDBM50410033(CHEMBL180120)
Affinity DataKi:  1.95E+3nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410029BDBM50410029(CHEMBL181507)
Affinity DataKi:  3.31E+3nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410030BDBM50410030(CHEMBL426424)
Affinity DataKi:  4.79E+3nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Clarkson University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410040BDBM50410040(CHEMBL179666)
Affinity DataKi:  7.94E+3nMAssay Description:Antiviral activity potency was assessed by measuring effect on the accumulation of viral RNA transcripts 3 days after infection of MT-2 cells with HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed