Compile Data Set for Download or QSAR
maximum 50k data
Found 55 Enz. Inhib. hit(s) with all data for entry = 50016510
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169847(4-(4-Azetidin-1-yl-benzenesulfonyl)-1-[2-(2,4-difl...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169848(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(3-fl...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169840(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(2-fl...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169842(1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophen...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108699(1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfony...)
Affinity DataKi:  0.420nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169846(2-(4-Benzenesulfonyl-piperidin-1-yl)-1-(2,4-difluo...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169842(1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophen...)
Affinity DataKi:  0.630nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169841(4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-ph...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169844(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-[1...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169838(4-Benzenesulfonyl-1-[2-(2,4-difluoro-phenyl)-ethyl...)
Affinity DataKi:  0.680nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169847(4-(4-Azetidin-1-yl-benzenesulfonyl)-1-[2-(2,4-difl...)
Affinity DataKi:  1nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169839(4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-pipe...)
Affinity DataKi:  1.33nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169845(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-py...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169845(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-py...)
Affinity DataKi:  2nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169846(2-(4-Benzenesulfonyl-piperidin-1-yl)-1-(2,4-difluo...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169839(4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-pipe...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169840(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(2-fl...)
Affinity DataKi:  14nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi:  25nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169838(4-Benzenesulfonyl-1-[2-(2,4-difluoro-phenyl)-ethyl...)
Affinity DataKi:  49nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169848(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(3-fl...)
Affinity DataKi:  49nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108699(1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfony...)
Affinity DataKi:  92nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169846(2-(4-Benzenesulfonyl-piperidin-1-yl)-1-(2,4-difluo...)
Affinity DataKi:  130nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169842(1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophen...)
Affinity DataKi:  176nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169840(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(2-fl...)
Affinity DataKi:  266nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169842(1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophen...)
Affinity DataKi:  313nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169841(4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-ph...)
Affinity DataKi:  397nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169841(4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-ph...)
Affinity DataKi:  398nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169840(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(2-fl...)
Affinity DataKi:  398nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108699(1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfony...)
Affinity DataKi:  710nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169848(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(3-fl...)
Affinity DataKi:  791nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169847(4-(4-Azetidin-1-yl-benzenesulfonyl)-1-[2-(2,4-difl...)
Affinity DataKi:  844nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169839(4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-pipe...)
Affinity DataKi:  863nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169838(4-Benzenesulfonyl-1-[2-(2,4-difluoro-phenyl)-ethyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169841(4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-ph...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169839(4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-pipe...)
Affinity DataKi:  1.49E+3nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169846(2-(4-Benzenesulfonyl-piperidin-1-yl)-1-(2,4-difluo...)
Affinity DataKi: >1.50E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108699(1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfony...)
Affinity DataKi: >1.50E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi: >1.50E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169848(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(3-fl...)
Affinity DataKi:  1.53E+3nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169847(4-(4-Azetidin-1-yl-benzenesulfonyl)-1-[2-(2,4-difl...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169845(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-py...)
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169844(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-[1...)
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity against human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169838(4-Benzenesulfonyl-1-[2-(2,4-difluoro-phenyl)-ethyl...)
Affinity DataKi:  2.45E+3nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169839(4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-pipe...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity against human IKr channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169844(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-[1...)
Affinity DataKi: >4.00E+3nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169845(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-py...)
Affinity DataKi: >4.00E+3nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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