Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50016544
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170292BDBM50170292((S)-2-{4'-[(5-Methanesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50: 0.430nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170302BDBM50170302((S)-2-{4'-[(5-Chloro-benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170287BDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 0.660nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170300BDBM50170300((S)-3-Methyl-2-{4'-[(5-nitro-benzofuran-2-carbonyl...)
Affinity DataIC50: 0.700nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170294BDBM50170294((S)-2-{4'-[(5-Acetylamino-benzofuran-2-carbonyl)-a...)
Affinity DataIC50: 0.980nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 28485BDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170304BDBM50170304((S)-2-{4'-[(5-Amino-benzofuran-2-carbonyl)-amino]-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170287BDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170287BDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170300BDBM50170300((S)-3-Methyl-2-{4'-[(5-nitro-benzofuran-2-carbonyl...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170299BDBM50170299((S)-3-Methyl-2-{4'-[([1,2,3]thiadiazole-4-carbonyl...)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170289BDBM50170289((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 2.20nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170298BDBM50170298((S)-2-{4'-[(4-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 2.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170295BDBM50170295((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 2.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170302BDBM50170302((S)-2-{4'-[(5-Chloro-benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50: 3.20nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170288BDBM50170288((S)-2-{4'-[(5-Benzenesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50: 3.40nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170296BDBM50170296((S)-2-{4'-[(4-Benzyloxy-benzofuran-2-carbonyl)-ami...)
Affinity DataIC50: 3.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170292BDBM50170292((S)-2-{4'-[(5-Methanesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170294BDBM50170294((S)-2-{4'-[(5-Acetylamino-benzofuran-2-carbonyl)-a...)
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrilysin(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 28485BDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataEC50:  4nMAssay Description:Inhibitory concentration against MMP-7More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170286BDBM50170286((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 4.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170301BDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50: 4.90nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 28485BDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170305BDBM50170305((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 8.10nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170289BDBM50170289((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 8.40nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170295BDBM50170295((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170299BDBM50170299((S)-3-Methyl-2-{4'-[([1,2,3]thiadiazole-4-carbonyl...)
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170291BDBM50170291((S)-2-{4'-[(7-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170303BDBM50170303((S)-2-[4'-(3-Methoxy-benzoylamino)-biphenyl-4-sulf...)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170303BDBM50170303((S)-2-[4'-(3-Methoxy-benzoylamino)-biphenyl-4-sulf...)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170293BDBM50170293((S)-2-(4'-{[4-(1-Carboxy-ethoxy)-benzofuran-2-carb...)
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170298BDBM50170298((S)-2-{4'-[(4-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 16nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170288BDBM50170288((S)-2-{4'-[(5-Benzenesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170297BDBM50170297((S)-2-{4'-[(1H-Indole-2-carbonyl)-amino]-biphenyl-...)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170291BDBM50170291((S)-2-{4'-[(7-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170290BDBM50170290({4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl-4-sul...)
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170301BDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50: 23nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170286BDBM50170286((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 28nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170297BDBM50170297((S)-2-{4'-[(1H-Indole-2-carbonyl)-amino]-biphenyl-...)
Affinity DataIC50: 35nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170305BDBM50170305((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50: 37nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170290BDBM50170290({4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl-4-sul...)
Affinity DataIC50: 47nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170296BDBM50170296((S)-2-{4'-[(4-Benzyloxy-benzofuran-2-carbonyl)-ami...)
Affinity DataIC50: 62nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170293BDBM50170293((S)-2-(4'-{[4-(1-Carboxy-ethoxy)-benzofuran-2-carb...)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 28485BDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149234BDBM50149234(N-(4-morpholinobutyl)benzofuran-2-carboxamide | Be...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170297BDBM50170297((S)-2-{4'-[(1H-Indole-2-carbonyl)-amino]-biphenyl-...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170301BDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Bovine)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149216BDBM50149216(WAY-170523 | Benzofuran-2-carboxylic acid (2-{4-[b...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170291BDBM50170291((S)-2-{4'-[(7-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170290BDBM50170290({4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl-4-sul...)
Affinity DataIC50: 1.39E+4nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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