Compile Data Set for Download or QSAR
maximum 50k data
Found 52 Enz. Inhib. hit(s) with all data for entry = 50016544
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170292((S)-2-{4'-[(5-Methanesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  0.430nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170302((S)-2-{4'-[(5-Chloro-benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  0.600nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  0.660nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170300((S)-3-Methyl-2-{4'-[(5-nitro-benzofuran-2-carbonyl...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170294((S)-2-{4'-[(5-Acetylamino-benzofuran-2-carbonyl)-a...)
Affinity DataIC50:  0.980nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170304((S)-2-{4'-[(5-Amino-benzofuran-2-carbonyl)-amino]-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170300((S)-3-Methyl-2-{4'-[(5-nitro-benzofuran-2-carbonyl...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170299((S)-3-Methyl-2-{4'-[([1,2,3]thiadiazole-4-carbonyl...)
Affinity DataIC50:  2.10nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170289((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170298((S)-2-{4'-[(4-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170295((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170302((S)-2-{4'-[(5-Chloro-benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170288((S)-2-{4'-[(5-Benzenesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170296((S)-2-{4'-[(4-Benzyloxy-benzofuran-2-carbonyl)-ami...)
Affinity DataIC50:  3.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170292((S)-2-{4'-[(5-Methanesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170294((S)-2-{4'-[(5-Acetylamino-benzofuran-2-carbonyl)-a...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170286((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50:  4.90nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170305((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  8.10nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170289((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  8.40nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170295((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170299((S)-3-Methyl-2-{4'-[([1,2,3]thiadiazole-4-carbonyl...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170291((S)-2-{4'-[(7-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170303((S)-2-[4'-(3-Methoxy-benzoylamino)-biphenyl-4-sulf...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170303((S)-2-[4'-(3-Methoxy-benzoylamino)-biphenyl-4-sulf...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170293((S)-2-(4'-{[4-(1-Carboxy-ethoxy)-benzofuran-2-carb...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170298((S)-2-{4'-[(4-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  16nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170297((S)-2-{4'-[(1H-Indole-2-carbonyl)-amino]-biphenyl-...)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170288((S)-2-{4'-[(5-Benzenesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170291((S)-2-{4'-[(7-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170290(CHEMBL189955 | {4'-[(Benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  22nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50:  23nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170286((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  28nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170297((S)-2-{4'-[(1H-Indole-2-carbonyl)-amino]-biphenyl-...)
Affinity DataIC50:  35nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170305((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  37nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170290(CHEMBL189955 | {4'-[(Benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  47nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170296((S)-2-{4'-[(4-Benzyloxy-benzofuran-2-carbonyl)-ami...)
Affinity DataIC50:  62nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170293((S)-2-(4'-{[4-(1-Carboxy-ethoxy)-benzofuran-2-carb...)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibitory concentration against MMP-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149234(Benzofuran-2-carboxylic acid (4-morpholin-4-yl-but...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170297((S)-2-{4'-[(1H-Indole-2-carbonyl)-amino]-biphenyl-...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149216(Benzofuran-2-carboxylic acid (2-{4-[benzyl-(2-hydr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170291((S)-2-{4'-[(7-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170290(CHEMBL189955 | {4'-[(Benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibitory concentration against MMP-14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50: >1.60E+4nMAssay Description:Inhibitory concentration against MMP-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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