Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50016556
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170625(3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50164243((R)-1-(3'-cyanobiphenyl-4-yl)-3-(4-fluoro-3-(trifl...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170614(1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperi...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170617(1-(3'-cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperi...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170622(3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170626(1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopropylmethyl-...)
Affinity DataKi:  4nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170613(1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoro...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170608(3-(3-Chloro-phenyl)-1-(3'-cyano-biphenyl-4-yl)-1-(...)
Affinity DataKi:  5.80nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170615(3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-...)
Affinity DataKi:  6nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170618(1-(3'-Cyano-biphenyl-4-yl)-1-(2-dimethylamino-ethy...)
Affinity DataKi:  6nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170630(1-(3'-Cyano-biphenyl-4-yl)-1-(1-ethyl-piperidin-4-...)
Affinity DataKi:  7.10nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170616(3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-...)
Affinity DataKi:  7.10nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170620(1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoro...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170624(1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoro...)
Affinity DataKi:  8.20nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170628(1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoro...)
Affinity DataKi:  8.90nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170611(1-(3'-Cyano-biphenyl-4-yl)-3-(3,4-dichloro-phenyl)...)
Affinity DataKi:  11nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170619(1-(3'-Chloro-biphenyl-4-yl)-1-(1-cyclopentyl-piper...)
Affinity DataKi:  12.5nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170612(1-(3'-Cyano-biphenyl-4-yl)-3-(3,4-dichloro-phenyl)...)
Affinity DataKi:  19nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170627(1-(1-Cyclopentyl-piperidin-4-yl)-3-(3,4-dichloro-p...)
Affinity DataKi:  20nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170621(1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperi...)
Affinity DataKi:  98nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170623(1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperi...)
Affinity DataKi:  139nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170631(1-(3'-Cyano-biphenyl-4-yl)-1-(1-ethanesulfonyl-pip...)
Affinity DataKi:  166nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170609(1-(1-Cyclopentyl-piperidin-4-yl)-3-(3,4-dichloro-p...)
Affinity DataKi:  197nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170629(1-(3'-Cyano-biphenyl-4-yl)-1-(1-cyclopentyl-piperi...)
Affinity DataKi:  233nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170610(1-(3'-Cyano-biphenyl-4-yl)-3-(4-fluoro-3-trifluoro...)
Affinity DataKi:  374nMAssay Description:Inhibition of human melanin concentrating hormone receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170624(1-(3'-Cyano-biphenyl-4-yl)-3-(3-fluoro-4-trifluoro...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptake by serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50170622(3-(3-Chloro-4-fluoro-phenyl)-1-(3'-cyano-biphenyl-...)
Affinity DataKi:  1.08E+3nMAssay Description:Inhibition of 5-hydroxytryptamine reuptake by serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed