Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50037521
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170788(CHEMBL410967 | Degarelix analogue)
Affinity DataIC50:  1.38nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50209591(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Atz)]-D-[Aph(...)
Affinity DataIC50:  1.40nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170789(CHEMBL265879 | Degarelix analogue)
Affinity DataIC50:  1.47nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170774(CHEMBL405273 | Degarelix analogue)
Affinity DataIC50:  1.5nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170770(CHEMBL428825 | Degarelix analogue)
Affinity DataIC50:  1.54nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170776(CHEMBL414347 | Degarelix analogue)
Affinity DataIC50:  1.56nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170798(CHEMBL413450 | Degarelix analogue)
Affinity DataIC50:  1.62nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102450(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(DHor)]-D-[Aph...)
Affinity DataIC50:  1.64nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170767(CHEMBL264090 | Degarelix analogue)
Affinity DataIC50:  1.72nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170791(CHEMBL415820 | Degarelix analogue)
Affinity DataIC50:  1.77nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170769(CHEMBL267873 | Degarelix analogue)
Affinity DataIC50:  1.77nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170779(CHEMBL415595 | Degarelix analogue)
Affinity DataIC50:  1.83nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170785(CHEMBL412500 | Degarelix analogue)
Affinity DataIC50:  1.85nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170768(CHEMBL265020 | Degarelix analogue)
Affinity DataIC50:  1.97nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170792(CHEMBL438905 | Degarelix analogue)
Affinity DataIC50:  1.98nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170795(CHEMBL441893 | Degarelix analogue)
Affinity DataIC50:  2.01nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170787(CHEMBL415622 | Degarelix analogue)
Affinity DataIC50:  2.11nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170797(CHEMBL402683 | Degarelix analogue)
Affinity DataIC50:  2.24nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170782(CHEMBL414507 | Degarelix analogue)
Affinity DataIC50:  2.71nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170780(CHEMBL437672 | Degarelix analogue)
Affinity DataIC50:  2.85nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170799(CHEMBL415549 | Degarelix analogue)
Affinity DataIC50:  3.5nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170790(CHEMBL414346 | Degarelix analogue)
Affinity DataIC50:  3.79nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170784(CHEMBL406225 | Degarelix analogue)
Affinity DataIC50:  4.25nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170783(CHEMBL266444 | Degarelix analogue)
Affinity DataIC50:  5.31nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170794(CHEMBL404973 | Degarelix analogue)
Affinity DataIC50:  5.52nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170771(CHEMBL429378 | Degarelix analogue)
Affinity DataIC50:  9.18nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170775(CHEMBL263507 | Degarelix analogue)
Affinity DataIC50:  10.6nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170777(CHEMBL415813 | Degarelix analogue)
Affinity DataIC50:  13.5nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170773(CHEMBL415328 | Degarelix analogue)
Affinity DataIC50:  22.6nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170796(CHEMBL268829 | Degarelix analogue)
Affinity DataIC50:  25.8nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170781(CHEMBL406535 | Degarelix analogue)
Affinity DataIC50:  48.9nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170786(CHEMBL266893 | Degarelix analogue)
Affinity DataIC50:  52.2nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170793(CHEMBL412212 | Degarelix analogue)
Affinity DataIC50:  178nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed