Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50037521
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170788(Degarelix analogue | CHEMBL410967)
Affinity DataIC50: 1.38nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50209591(Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Atz)]-D-[Aph(...)
Affinity DataIC50: 1.40nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170789(Degarelix analogue | CHEMBL265879)
Affinity DataIC50: 1.47nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170774(Degarelix analogue | CHEMBL405273)
Affinity DataIC50: 1.5nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170770(Degarelix analogue | CHEMBL428825)
Affinity DataIC50: 1.54nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170776(Degarelix analogue | CHEMBL414347)
Affinity DataIC50: 1.56nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170798(Degarelix analogue | CHEMBL413450)
Affinity DataIC50: 1.62nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50102450(degarelix | Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(D...)
Affinity DataIC50: 1.64nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170767(Degarelix analogue | CHEMBL264090)
Affinity DataIC50: 1.72nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170791(Degarelix analogue | CHEMBL415820)
Affinity DataIC50: 1.77nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170769(Degarelix analogue | CHEMBL267873)
Affinity DataIC50: 1.77nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170779(Degarelix analogue | CHEMBL415595)
Affinity DataIC50: 1.83nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170785(Degarelix analogue | CHEMBL412500)
Affinity DataIC50: 1.85nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170768(Degarelix analogue | CHEMBL265020)
Affinity DataIC50: 1.97nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170792(Degarelix analogue | CHEMBL438905)
Affinity DataIC50: 1.98nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170795(Degarelix analogue | CHEMBL441893)
Affinity DataIC50: 2.01nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170787(Degarelix analogue | CHEMBL415622)
Affinity DataIC50: 2.11nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170797(Degarelix analogue | CHEMBL402683)
Affinity DataIC50: 2.24nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170782(Degarelix analogue | CHEMBL414507)
Affinity DataIC50: 2.71nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170780(Degarelix analogue | CHEMBL437672)
Affinity DataIC50: 2.85nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170799(Degarelix analogue | CHEMBL415549)
Affinity DataIC50: 3.5nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170790(Degarelix analogue | CHEMBL414346)
Affinity DataIC50: 3.79nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170784(Degarelix analogue | CHEMBL406225)
Affinity DataIC50: 4.25nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170783(Degarelix analogue | CHEMBL266444)
Affinity DataIC50: 5.31nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170794(Degarelix analogue | CHEMBL404973)
Affinity DataIC50: 5.52nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170771(Degarelix analogue | CHEMBL429378)
Affinity DataIC50: 9.18nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170775(Degarelix analogue | CHEMBL263507)
Affinity DataIC50: 10.6nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170777(Degarelix analogue | CHEMBL415813)
Affinity DataIC50: 13.5nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170773(Degarelix analogue | CHEMBL415328)
Affinity DataIC50: 22.6nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170796(Degarelix analogue | CHEMBL268829)
Affinity DataIC50: 25.8nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170781(Degarelix analogue | CHEMBL406535)
Affinity DataIC50: 48.9nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170786(Degarelix analogue | CHEMBL266893)
Affinity DataIC50: 52.2nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50170793(Degarelix analogue | CHEMBL412212)
Affinity DataIC50: 178nMAssay Description:Antagonism of GnRH response in HEK293 cells expressing human GnRH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed