Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50016663
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50164279((S)-3-(aminomethyl)-5-methylhexanoic acid | (S)-3-...)
Affinity DataIC50:  73nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171790((S)-3-(aminomethyl)-4-(furan-2-yl)butanoic acid | ...)
Affinity DataIC50:  178nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171795(3-(aminomethyl)-4-(furan-2-yl)butanoic acid | CHEM...)
Affinity DataIC50:  421nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171794(3-(aminomethyl)-4-(furan-3-yl)butanoic acid | CHEM...)
Affinity DataIC50:  518nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171796(3-(aminomethyl)-4-(thiophen-3-yl)butanoic acid | C...)
Affinity DataIC50:  832nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171792((R)-3-(aminomethyl)-4-(furan-2-yl)butanoic acid | ...)
Affinity DataIC50:  1.46E+3nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171789(3-(aminomethyl)-4-(thiophen-2-yl)butanoic acid | C...)
Affinity DataIC50:  2.14E+3nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171791(3-(aminomethyl)-4-phenylbutanoic acid | CHEMBL2061...)
Affinity DataIC50: >1.00E+7nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel alpha-2 delta subunit(Sus scrofa)
Pgrd Michigan Laboratories

Curated by ChEMBL
LigandPNGBDBM50171793(3-(aminomethyl)-4-(tetrahydrofuran-3-yl)butanoic a...)
Affinity DataIC50: >1.00E+7nMAssay Description:Displacement of [3H]gabapentin from alpha2delta calcium channel in pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed