Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50037599
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataIC50: 0.430nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173859(Diphenylmethoxypiperidine derivative | CHEMBL37062...)
Affinity DataIC50: 12.5nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173856(4-[bis(4-fluorophenyl)methoxy]-1-methylpiperidine ...)
Affinity DataIC50: 22.1nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173854((RS )-(+/-)-4-(Bis-(4-chlorophenyl)methoxy)-1-meth...)
Affinity DataIC50: 44nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173853(Diphenylmethoxypiperidine derivative | CHEMBL38124...)
Affinity DataIC50: 50.6nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50084717(CHEMBL120901 | 3-Naphthalen-2-yl-8-oxa-bicyclo[3.2...)
Affinity DataIC50: 104nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173860(4-[(4-chlorophenyl)(phenyl)methoxy]-1-methylpiperi...)
Affinity DataIC50: 155nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173861(4-[1-(4-fluorophenyl)ethoxy]-1-methylpiperidine | ...)
Affinity DataIC50: 264nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173855(4-[(4-fluorophenyl)(phenyl)methoxy]-1-methylpiperi...)
Affinity DataIC50: 277nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50173858(1-methyl-4-[(3-methylphenyl)(phenyl)methoxy]piperi...)
Affinity DataIC50: 293nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wake Forest University Health Sciences

Curated by ChEMBL
LigandPNGBDBM50241333(4-(benzhydryloxy)-1-methylpiperidine | CHEMBL1492 ...)
Affinity DataIC50: 420nMAssay Description:Displacement of [125I]RTI-55 dopamine transporter binding in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed