Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 2575
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22218(1-[(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-o...)
Affinity DataIC50: 0.300nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22220(1-{[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-...)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22215(1-({4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-y...)
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22218(1-[(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-o...)
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22219(1-{[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-...)
Affinity DataIC50: 0.5nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22215(1-({4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-y...)
Affinity DataIC50: 0.5nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22209(1-[(4-{5-[4-(2-methylpropyl)phenyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 0.600nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22220(1-{[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-...)
Affinity DataIC50: 0.800nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22216(1-({4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 0.800nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22219(1-{[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-...)
Affinity DataIC50: 0.900nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22209(1-[(4-{5-[4-(2-methylpropyl)phenyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 1nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22205(1-[(4-{5-[4-(2-methylbutan-2-yl)phenyl]-1,2,4-oxad...)
Affinity DataIC50: 1.30nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22206(1-({4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 1.30nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22216(1-({4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 1.40nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22206(1-({4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 1.60nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22217(1-({4-[5-(4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 1.70nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22212(1-[(4-{5-[4-(propan-2-yloxy)phenyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 1.80nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22205(1-[(4-{5-[4-(2-methylbutan-2-yl)phenyl]-1,2,4-oxad...)
Affinity DataIC50: 1.80nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22214(1-({4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 2.20nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22207(1-({4-[5-(4-butylphenyl)-1,2,4-oxadiazol-3-yl]phen...)
Affinity DataIC50: 2.40nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22207(1-({4-[5-(4-butylphenyl)-1,2,4-oxadiazol-3-yl]phen...)
Affinity DataIC50: 2.90nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22210(1-[(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxad...)
Affinity DataIC50: 3.80nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22204(1-({4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 3.80nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22214(1-({4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 4nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22213(1-({4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-y...)
Affinity DataIC50: 4.5nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22211(1-({4-[5-(4-ethoxyphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 5.10nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22204(1-({4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 5.20nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22208(1-({4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]phen...)
Affinity DataIC50: 6.40nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22210(1-[(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxad...)
Affinity DataIC50: 6.60nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22203(1-{4-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]...)
Affinity DataIC50: 8.20nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22217(1-({4-[5-(4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 11nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22212(1-[(4-{5-[4-(propan-2-yloxy)phenyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 12nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22213(1-({4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-y...)
Affinity DataIC50: 12nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22203(1-{4-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]...)
Affinity DataIC50: 20nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22221(2-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]ani...)
Affinity DataIC50: 27nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22208(1-({4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]phen...)
Affinity DataIC50: 29nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22216(1-({4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 40nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Merck Research Laboratories

LigandPNGBDBM22211(1-({4-[5-(4-ethoxyphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 48nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22215(1-({4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-y...)
Affinity DataIC50: 49nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22219(1-{[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-...)
Affinity DataIC50: 68nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22209(1-[(4-{5-[4-(2-methylpropyl)phenyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 70nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22205(1-[(4-{5-[4-(2-methylbutan-2-yl)phenyl]-1,2,4-oxad...)
Affinity DataIC50: 75nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22220(1-{[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-...)
Affinity DataIC50: 89nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22210(1-[(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxad...)
Affinity DataIC50: 90nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Merck Research Laboratories

LigandPNGBDBM22201(1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22206(1-({4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 150nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22217(1-({4-[5-(4-phenylphenyl)-1,2,4-oxadiazol-3-yl]phe...)
Affinity DataIC50: 240nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22207(1-({4-[5-(4-butylphenyl)-1,2,4-oxadiazol-3-yl]phen...)
Affinity DataIC50: 350nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22204(1-({4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 370nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Merck Research Laboratories

LigandPNGBDBM22212(1-[(4-{5-[4-(propan-2-yloxy)phenyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 370nMT: 2°CAssay Description:The assay measures the displacement of [33P]-labeled sphingosine-1-phosphate (S1P) by test compounds from human S1P receptors expressed on CHO cell m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2008
Entry Details Article
PubMed
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