Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50017027
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against PDE2 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 635nMAssay Description:Inhibitory activity against PDE2 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibitory activity against PDE11 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE8B by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE9 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE10 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE11 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE3 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4B by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE8B by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE3 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4A by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE5 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE9 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4A by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE5 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4B by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE8A by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4D by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4C by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4C by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50176521(5-methyl-6-oxo-6,7-dihydro-5H-furo[2,3-f]indole-7-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE10 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE4D by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28393((2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol | CHEM...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against PDE8A by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed