Compile Data Set for Download or QSAR
maximum 50k data
Found 61 Enz. Inhib. hit(s) with all data for entry = 50017049
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(CHEMBL224545 | methyl 4-(4-methoxyphenethylamino)-...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(CHEMBL224545 | methyl 4-(4-methoxyphenethylamino)-...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(CHEMBL224545 | methyl 4-(4-methoxyphenethylamino)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in presence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in presence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176835(CHEMBL223871 | ethyl 4-(4-methoxyphenethylamino)-1...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176815(CHEMBL225398 | ethyl 4-(4-fluorophenethylamino)-1-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176838(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176842(CHEMBL224620 | ethyl 4-(2-fluorophenethylamino)-1-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176815(CHEMBL225398 | ethyl 4-(4-fluorophenethylamino)-1-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176822(CHEMBL375154 | isopropyl 4-(4-methoxyphenethylamin...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176832(CHEMBL224909 | ethyl 4-(4-chlorophenethylamino)-1-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176855(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176844(CHEMBL389405 | isopropyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176835(CHEMBL223871 | ethyl 4-(4-methoxyphenethylamino)-1...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176842(CHEMBL224620 | ethyl 4-(2-fluorophenethylamino)-1-...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176849(CHEMBL427255 | isopropyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176828(CHEMBL224097 | ethyl 4-(3-fluorophenethylamino)-1-...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176840(CHEMBL224083 | isopropyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176825(CHEMBL389060 | isopropyl 4-(4-chlorophenethylamino...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176839(CHEMBL223821 | isopropyl 4-(2-chlorophenethylamino...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176848(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176834(CHEMBL224307 | cyclopropylmethyl 1-(2-chloro-2-phe...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176850(CHEMBL223450 | sec-butyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176843(CHEMBL374620 | sec-butyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176852(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176847(CHEMBL224313 | ethyl 4-(2-chlorophenethylamino)-1-...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176830(CHEMBL391004 | methyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176833(CHEMBL224545 | methyl 4-(4-methoxyphenethylamino)-...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176845(CHEMBL224619 | isopropyl 4-(3-chlorophenethylamino...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176820(4-butyl-5-(4-cyclopropylbut-1-en-2-yl)-1-(2-phenyl...)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176826(CHEMBL390096 | propyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176819(CHEMBL225026 | methyl 4-(benzylamino)-1-(2-chloro-...)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176818(CHEMBL223451 | propyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176838(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176832(CHEMBL224909 | ethyl 4-(4-chlorophenethylamino)-1-...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176831(CHEMBL376193 | propyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176836(CHEMBL225341 | methyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176841(CHEMBL389644 | ethyl 4-(3-chlorophenethylamino)-1-...)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176853(CHEMBL224852 | sec-butyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176816(CHEMBL224669 | methyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176851(CHEMBL224098 | isopropyl 4-(benzylamino)-1-(2-chlo...)
Affinity DataKi:  559nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176827(CHEMBL223229 | butyl 1-(2-chloro-2-phenylethyl)-4-...)
Affinity DataKi:  895nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176846(CHEMBL376747 | butyl 1-(2-chloro-2-phenylethyl)-4-...)
Affinity DataKi:  959nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176823(CHEMBL224621 | isopropyl 1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176830(CHEMBL391004 | methyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176826(CHEMBL390096 | propyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50176854(CHEMBL224179 | propyl 4-(benzylamino)-1-(2-chloro-...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50176818(CHEMBL223451 | propyl 1-(2-chloro-2-phenylethyl)-4...)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 61 total ) | Next | Last >>
Jump to: