Compile Data Set for Download or QSAR
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Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50017184
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178759(1,6-bis-(N,N-dimethyl-Dmt-Tic-NH)hexane | CHEMBL37...)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178757(3-(Dmt-Tic-NH-butyl)-6-(Dmt-Tic-NH-propyl)-2-(1H)-...)
Affinity DataKi:  0.0920nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178761(3,6-bis(Dmt-Tic-NH-ethyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataKi:  0.0950nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178756(3-(Dmt-Tic-NH-ethyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-p...)
Affinity DataKi:  0.107nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178765(1,4-bis-(Dmt-Tic-amino)butane | CHEMBL370197)
Affinity DataKi:  0.124nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178762(1,6-bis-(Dmt-Tic-amino)hexane | CHEMBL197185)
Affinity DataKi:  0.129nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178763(3,6-bis(Dmt-Tic-NH-propyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataKi:  0.155nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178764(3-(Dmt-Tic-NH-propyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178755(3,6-bis(Dmt-Tic-NH-methyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataKi:  0.163nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178754(3,6-bis-(N,N-dimethyl-Dmt-Tic-NH-propyl)-2(1H)-pyr...)
Affinity DataKi:  0.287nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178758(3,6-bis(Dmt-Tic-NH-butyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataKi:  0.323nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178756(3-(Dmt-Tic-NH-ethyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-p...)
Affinity DataKi:  1.37nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178760(1,10-bis-(Dmt-Tic-amino)decane | CHEMBL373192)
Affinity DataKi:  1.53nMAssay Description:Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178764(3-(Dmt-Tic-NH-propyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-...)
Affinity DataKi:  1.56nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178754(3,6-bis-(N,N-dimethyl-Dmt-Tic-NH-propyl)-2(1H)-pyr...)
Affinity DataKi:  1.68nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178758(3,6-bis(Dmt-Tic-NH-butyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataKi:  1.74nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178762(1,6-bis-(Dmt-Tic-amino)hexane | CHEMBL197185)
Affinity DataKi:  1.79nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178759(1,6-bis-(N,N-dimethyl-Dmt-Tic-NH)hexane | CHEMBL37...)
Affinity DataKi:  2.21nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178757(3-(Dmt-Tic-NH-butyl)-6-(Dmt-Tic-NH-propyl)-2-(1H)-...)
Affinity DataKi:  2.28nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178761(3,6-bis(Dmt-Tic-NH-ethyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataKi:  2.83nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178763(3,6-bis(Dmt-Tic-NH-propyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataKi:  3.08nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178755(3,6-bis(Dmt-Tic-NH-methyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataKi:  3.76nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178760(1,10-bis-(Dmt-Tic-amino)decane | CHEMBL373192)
Affinity DataKi:  4.86nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178765(1,4-bis-(Dmt-Tic-amino)butane | CHEMBL370197)
Affinity DataKi:  5.72nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178762(1,6-bis-(Dmt-Tic-amino)hexane | CHEMBL197185)
Affinity DataIC50:  2.72E+3nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178760(1,10-bis-(Dmt-Tic-amino)decane | CHEMBL373192)
Affinity DataIC50:  5.43E+3nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178763(3,6-bis(Dmt-Tic-NH-propyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataIC50:  7.03E+3nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178763(3,6-bis(Dmt-Tic-NH-propyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178762(1,6-bis-(Dmt-Tic-amino)hexane | CHEMBL197185)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178754(3,6-bis-(N,N-dimethyl-Dmt-Tic-NH-propyl)-2(1H)-pyr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178758(3,6-bis(Dmt-Tic-NH-butyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178759(1,6-bis-(N,N-dimethyl-Dmt-Tic-NH)hexane | CHEMBL37...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178765(1,4-bis-(Dmt-Tic-amino)butane | CHEMBL370197)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178764(3-(Dmt-Tic-NH-propyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178755(3,6-bis(Dmt-Tic-NH-methyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178765(1,4-bis-(Dmt-Tic-amino)butane | CHEMBL370197)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178756(3-(Dmt-Tic-NH-ethyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178758(3,6-bis(Dmt-Tic-NH-butyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178757(3-(Dmt-Tic-NH-butyl)-6-(Dmt-Tic-NH-propyl)-2-(1H)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178761(3,6-bis(Dmt-Tic-NH-ethyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178764(3-(Dmt-Tic-NH-propyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178760(1,10-bis-(Dmt-Tic-amino)decane | CHEMBL373192)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178757(3-(Dmt-Tic-NH-butyl)-6-(Dmt-Tic-NH-propyl)-2-(1H)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178755(3,6-bis(Dmt-Tic-NH-methyl)-2(1H)-pyrazinone | CHEM...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at mu opioid receptor in myenteric plexus longitudinal muscle of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178756(3-(Dmt-Tic-NH-ethyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178754(3,6-bis-(N,N-dimethyl-Dmt-Tic-NH-propyl)-2(1H)-pyr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178759(1,6-bis-(N,N-dimethyl-Dmt-Tic-NH)hexane | CHEMBL37...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50178761(3,6-bis(Dmt-Tic-NH-ethyl)-2(1H)-pyrazinone | CHEMB...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed