Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50017248
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179600BDBM50179600(5-(2-fluorobenzylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50: 40nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179631BDBM50179631(5-(sec-butylthio)-1-(5-(methylsulfonyl)pyridin-2-y...)
Affinity DataIC50: 50nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179598BDBM50179598(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(propylthio)-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179609BDBM50179609(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(phenylthio)-...)
Affinity DataIC50: 60nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179596BDBM50179596(5-(cyclopentylmethoxy)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50: 60nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179611BDBM50179611(5-(cycloheptyloxy)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50: 70nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179616BDBM50179616(5-(benzylthio)-1-(5-(methylsulfonyl)pyridin-2-yl)-...)
Affinity DataIC50: 80nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179606BDBM50179606(5-(cyclobutylmethoxy)-1-(5-(methylsulfonyl)pyridin...)
Affinity DataIC50: 80nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179620BDBM50179620(5-((4-methylenecyclohexyl)methoxy)-1-(5-(methylsul...)
Affinity DataIC50: 90nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179591BDBM50179591(5-(3-methylbutan-2-yloxy)-1-(5-(methylsulfonyl)pyr...)
Affinity DataIC50: 90nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179621BDBM50179621(5-(cyclohexylthio)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179624BDBM50179624(5-(2,3-dimethylphenoxy)-1-(5-(methylsulfonyl)pyrid...)
Affinity DataIC50: 100nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179602BDBM50179602(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(5,6,7,8-tetr...)
Affinity DataIC50: 100nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179592BDBM50179592(5-isobutoxy-1-(5-(methylsulfonyl)pyridin-2-yl)-3-(...)
Affinity DataIC50: 110nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179601BDBM50179601(5-(cyclohex-3-enylmethoxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50: 140nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50176545BDBM50176545(3-(difluoromethyl)-5-((2R,6S)-2,6-dimethylmorpholi...)
Affinity DataIC50: 140nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179595BDBM50179595(5-(3-methylcyclopentyloxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50: 160nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179624BDBM50179624(5-(2,3-dimethylphenoxy)-1-(5-(methylsulfonyl)pyrid...)
Affinity DataIC50: 170nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179608BDBM50179608(5-(2-ethoxyethylthio)-1-(5-(methylsulfonyl)pyridin...)
Affinity DataIC50: 170nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179610BDBM50179610(5-(2-methylpentan-3-yloxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50: 170nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179609BDBM50179609(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(phenylthio)-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179598BDBM50179598(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(propylthio)-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179593BDBM50179593(5-(2-methylcyclohexyloxy)-1-(5-(methylsulfonyl)pyr...)
Affinity DataIC50: 200nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179625BDBM50179625(5-(cyclopentyloxy)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50: 210nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179628BDBM50179628(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(pentylthio)-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50137425BDBM50137425(2-(3-Difluoromethyl-5-phenyl-pyrazol-1-yl)-5-metha...)
Affinity DataIC50: 310nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179613BDBM50179613(5-(4-methylpentylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50: 400nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179596BDBM50179596(5-(cyclopentylmethoxy)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50: 400nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024426BDBM50024426(CHEMBL204252)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179599BDBM50179599(2-(4-methyl-5-(pentan-3-yloxy)-3-(trifluoromethyl)...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179603BDBM50179603(2-(5-(cyclopentyloxy)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179605BDBM50179605(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(pentan-2-ylo...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179623BDBM50179623(5-(1-methoxybutan-2-yloxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179626BDBM50179626(2-(5-(cyclohexyloxy)-3-(trifluoromethyl)-1H-pyrazo...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179607BDBM50179607(2-(5-(benzyloxy)-3-(trifluoromethyl)-1H-pyrazol-1-...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179629BDBM50179629(1-(5-(methylsulfonyl)pyridin-2-yl)-5-phenoxy-3-(tr...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179630BDBM50179630(2-(5-(3-fluorobenzyloxy)-3-(trifluoromethyl)-1H-py...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179633BDBM50179633(2-(4-chloro-5-isopropoxy-3-(trifluoromethyl)-1H-py...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179612BDBM50179612(2-(5-butoxy-3-(trifluoromethyl)-1H-pyrazol-1-yl)-5...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179614BDBM50179614(5-(methylsulfonyl)-2-(5-(pyridin-4-ylmethoxy)-3-(t...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179632BDBM50179632(2-(5-methoxy-3-(trifluoromethyl)-1H-pyrazol-1-yl)-...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179617BDBM50179617(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(tetrahydrofu...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179634BDBM50179634(2-(5-isopropoxy-3-(trifluoromethyl)-1H-pyrazol-1-y...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179594BDBM50179594(5-(methylsulfonyl)-2-(5-(naphthalen-1-ylmethoxy)-3...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179597BDBM50179597(2-(5-(cyclopropylmethoxy)-3-(trifluoromethyl)-1H-p...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179618BDBM50179618(2-(5-isobutoxy-4-methyl-3-(trifluoromethyl)-1H-pyr...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179619BDBM50179619(2-(5-isopropoxy-4-methyl-3-(trifluoromethyl)-1H-py...)
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179622BDBM50179622(5-cyclobutoxy-1-(5-(methylsulfonyl)pyridin-2-yl)-3...)
Affinity DataIC50: 550nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179600BDBM50179600(5-(2-fluorobenzylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50: 600nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Dog)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179602BDBM50179602(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(5,6,7,8-tetr...)
Affinity DataIC50: 900nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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