Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50017254
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179750BDBM50179750((S)-2-((S)-2-(benzyloxycarbonyl)-4-methylpentanami...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179749BDBM50179749((S)-2-(2-(2-(10H-phenothiazin-2-yloxy)acetamido)ac...)
Affinity DataIC50: 8nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179745BDBM50179745((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50: 25nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179747BDBM50179747((S)-2-((2S,3S)-2-(2-(10H-phenothiazin-2-yloxy)acet...)
Affinity DataIC50: 38nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179743BDBM50179743((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50: 48.7nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179744BDBM50179744((S)-4-Methyl-2-[(S)-4-methyl-2-(2-10H-phenothiazin...)
Affinity DataIC50: 55.4nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179741BDBM50179741((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50: 75.9nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179738BDBM50179738(N-((S)-1-((S)-1-((3S)-2-hydroxy-tetrahydrofuran-3-...)
Affinity DataIC50: 85.5nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179746BDBM50179746((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50: 88.6nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179739BDBM50179739((S)-4-Methyl-2-{(S)-4-methyl-2-[2-(10H-phenothiazi...)
Affinity DataIC50: 105nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179754BDBM50179754((S)-2-(2-(2-(10H-phenothiazin-2-yloxy)acetamido)-2...)
Affinity DataIC50: 138nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179748BDBM50179748((S)-4-methyl-2-[(S)-4-methyl-2-(3-10H-phenothiazin...)
Affinity DataIC50: 150nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179753BDBM50179753((S)-4-Methyl-2-{(S)-2-[2-(10H-phenothiazin-2-yloxy...)
Affinity DataIC50: 151nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179740BDBM50179740((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50: 222nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179751BDBM50179751((S)-2-((S)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50: 354nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179752BDBM50179752((S)-2-((R)-2-(2-(10H-phenothiazin-2-yloxy)acetamid...)
Affinity DataIC50: 553nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain small subunit 1/1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179742BDBM50179742((3S)-3-((S)-4-methyl-2-((S)-4-methyl-2-(10H-phenot...)
Affinity DataIC50: 905nMAssay Description:Inhibition of isolated human calpain1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed