Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50017265
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179883((4-Isopropylphenyl)-(4-isoquinolin-5-yl-phthalazin...)
Affinity DataIC50:  17nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179881((4-Chlorophenyl)-(4-isoquinolin-5-yl-phthalazin-1-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179890((4-tert-Butylphenyl)-(4-isoquinolin-5-yl-phthalazi...)
Affinity DataIC50:  75nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179889(CHEMBL382818 | N-(4-(chlorodifluoromethoxy)phenyl)...)
Affinity DataIC50:  79nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179888((3,4-Dichloro-phenyl)-(4-isoquinolin-5-yl-phthalaz...)
Affinity DataIC50:  110nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179891((4-Chloro-3-trifluoromethylphenyl)-(4-isoquinolin-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179893((4-Isoquinolin-5-yl-phthalazin-1-yl)-(2-methyl-1Hi...)
Affinity DataIC50:  230nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179884((4-Isoquinolin-5-yl-phthalazin-1-yl)-m-tolylamine ...)
Affinity DataIC50:  270nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179894((4-Isoquinolin-5-yl-phthalazin-1-yl)-(4-morpholin-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179882((2-Fluoro-4-methylphenyl)-(4-isoquinolin-5-ylphtha...)
Affinity DataIC50:  430nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179886((4-tert-Butylphenyl)-(4-quinolin-5-yl-phthalazin-1...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179892(CHEMBL204053 | N-(4-chlorophenyl)-4-(1H-pyrazol-4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179885(CHEMBL208513 | N-(4-chlorophenyl)-4-(1-methyl-1H-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179895((4-Isoquinolin-5-yl-phthalazin-1-yl)-o-tolylamine ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179887((4-Chlorophenyl)-(4-quinolin-5-yl-phthalazin-1-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed