Compile Data Set for Download or QSAR
Report error Found 113 Enz. Inhib. hit(s) with all data for entry = 50017297
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50133231((R)-2-(4-iodo-2,5-dimethoxyphenyl)-1-methylethylam...)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180255(1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol | C...)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataIC50: 0.580nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50133231((R)-2-(4-iodo-2,5-dimethoxyphenyl)-1-methylethylam...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180258(1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol | C...)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180253(1-((S)-2-aminopropyl)-7-methyl-1H-indazol-6-ol | C...)
Affinity DataIC50: 0.740nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180257(1-(2-aminoethyl)-1H-indazol-6-ol | CHEMBL199385)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataIC50: 0.940nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180258(1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol | C...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180255(1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol | C...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180252((S)-2-(6-methoxyindazol-1-yl)-1-methylethylamine |...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180254(1-((S)-2-aminopropyl)-7-iodo-1H-indazol-6-ol | CHE...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180258(1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol | C...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014945(alpha-methyl-5-HT | alpha-methyl-5-hydroxytryptami...)
Affinity DataEC50:  1.80nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180253(1-((S)-2-aminopropyl)-7-methyl-1H-indazol-6-ol | C...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180252((S)-2-(6-methoxyindazol-1-yl)-1-methylethylamine |...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014219(CHEMBL31115 | 5-methoxy-alpha-methyltryptamine | 2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataEC50:  2nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180256(1-((R)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL4373...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014219(CHEMBL31115 | 5-methoxy-alpha-methyltryptamine | 2...)
Affinity DataEC50:  2.70nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  2.80nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014219(CHEMBL31115 | 5-methoxy-alpha-methyltryptamine | 2...)
Affinity DataEC50:  3.10nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  3.5nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014945(alpha-methyl-5-HT | alpha-methyl-5-hydroxytryptami...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180253(1-((S)-2-aminopropyl)-7-methyl-1H-indazol-6-ol | C...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataEC50:  3.70nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180255(1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol | C...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50133231((R)-2-(4-iodo-2,5-dimethoxyphenyl)-1-methylethylam...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180252((S)-2-(6-methoxyindazol-1-yl)-1-methylethylamine |...)
Affinity DataEC50:  4.20nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014945(alpha-methyl-5-HT | alpha-methyl-5-hydroxytryptami...)
Affinity DataEC50:  4.20nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180257(1-(2-aminoethyl)-1H-indazol-6-ol | CHEMBL199385)
Affinity DataEC50:  4.5nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014219(CHEMBL31115 | 5-methoxy-alpha-methyltryptamine | 2...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180254(1-((S)-2-aminopropyl)-7-iodo-1H-indazol-6-ol | CHE...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180255(1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol | C...)
Affinity DataEC50:  4.90nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180258(1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol | C...)
Affinity DataEC50:  5.5nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180258(1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol | C...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180255(1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol | C...)
Affinity DataEC50:  5.90nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180254(1-((S)-2-aminopropyl)-7-iodo-1H-indazol-6-ol | CHE...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180258(1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol | C...)
Affinity DataEC50:  6.10nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180252((S)-2-(6-methoxyindazol-1-yl)-1-methylethylamine |...)
Affinity DataEC50:  6.70nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014945(alpha-methyl-5-HT | alpha-methyl-5-hydroxytryptami...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180253(1-((S)-2-aminopropyl)-7-methyl-1H-indazol-6-ol | C...)
Affinity DataEC50:  7.30nMAssay Description:Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180252((S)-2-(6-methoxyindazol-1-yl)-1-methylethylamine |...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014219(CHEMBL31115 | 5-methoxy-alpha-methyltryptamine | 2...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataKi:  8.10nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50014219(CHEMBL31115 | 5-methoxy-alpha-methyltryptamine | 2...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180257(1-(2-aminoethyl)-1H-indazol-6-ol | CHEMBL199385)
Affinity DataEC50:  8.60nMAssay Description:Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 113 total ) | Next | Last >>
Jump to: