Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50017342
LigandChemical structure of BindingDB Monomer ID 50180775BDBM50180775([Aib29,Asp31,Pro34,Phe35]CGRP(27-37) | FV-Aib-TDVG...)
Affinity DataKi:  0.00200nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180778BDBM50180778(FV-Hyp-TDVGPFAF | CHEMBL2371891)
Affinity DataKi:  0.00600nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50062162BDBM50062162(FVPTDVGPFAF | CHEMBL264010)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180781BDBM50180781(FV-Tic-TDVGPFAF | CHEMBL2371890)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180777BDBM50180777(FV((1R,2R,3R)-beta-aminocyclopropane carboxylic ac...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180776BDBM50180776(FVPTDVG-Tic-FAF-Tic | CHEMBL2371892)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180776BDBM50180776(FVPTDVG-Tic-FAF-Tic | CHEMBL2371892)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I-Tyr10] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180783BDBM50180783(FVATDVGPFAF | CHEMBL385986)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50062214BDBM50062214(FVPTDVGAFAF | CHEMBL406459)
Affinity DataKi:  14nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50062162BDBM50062162(FVPTDVGPFAF | CHEMBL264010)
Affinity DataKi:  14nMAssay Description:Displacement of [125I-Tyr10] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50062214BDBM50062214(FVPTDVGAFAF | CHEMBL406459)
Affinity DataKi:  77nMAssay Description:Displacement of [125I-Tyr10] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180784BDBM50180784(FV-Hop-TDVGPFAF | CHEMBL2371889)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180785BDBM50180785(FVPTDVG((1S,2S,3S)-beta-aminocyclopropane carboxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180774BDBM50180774(FV((1S,2S,3S)-beta-aminocyclopropane carboxylic ac...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180779BDBM50180779(FVPTNVG((1R,2R,3R)-beta-aminocyclopropane carboxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180780BDBM50180780(FVPTNVG((1S,2S,3S)-beta-aminocyclopropane carboxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50180782BDBM50180782(FVPTDVG((1R,2R,3R)-beta-aminocyclopropane carboxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed