Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50017348
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180899({4-[4-(4-bromophenoxy)benzoyl]phenyl}acetic acid |...)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180895(4-(4-phenoxybenzoyl)phenylacetic acid | CHEMBL3700...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180893((3-methyl-4-(4-phenoxybenzoyl)phenyl)acetic acid |...)
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180898((3-fluoro-4-(4-phenoxybenzoyl)phenyl)acetic acid |...)
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180894(4-(4-Phenoxy-benzoyl)-benzoic acid | 4-(4-phenoxyb...)
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180896(4-(4-{[2,5-bis(trifluoromethyl)benzyl]oxy}benzoyl)...)
Affinity DataIC50: 113nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180901(4-[4-benzyloxy)benzoyl]benzoic acid | CHEMBL202871)
Affinity DataIC50: 119nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180902(4-[3-(benzyloxy)benzoyl]benzoic acid | CHEMBL38264...)
Affinity DataIC50: 131nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180903((E)-3-(4-(4-phenoxybenzoyl)phenyl)acrylic acid | C...)
Affinity DataIC50: 470nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180897(4-[4-(benzhydryloxy)benzoyl]benzoic acid | CHEMBL2...)
Affinity DataIC50: 790nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180893((3-methyl-4-(4-phenoxybenzoyl)phenyl)acetic acid |...)
Affinity DataIC50: 1.45E+3nMpH: 6.6Assay Description:Displacement of [3H]androstenedione from 5-alpha reductase1 in rat ventral prostrate homogenate at pH 6.6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50180900(3-[4-(4-phenoxybenzoyl)phenyl]propanoic acid | CHE...)
Affinity DataIC50: 2.80E+3nMAssay Description:Displacement of [3H]-[1-beta,2beta]-testosterone from 5alpha reductase2 in human prostrate homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed