Affinity DataKi: 0.580nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.15E+3nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.58E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair