Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 1167
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9543BDBM9543(N-[4-(chlorodifluoromethoxy)phenyl]-5-{2-[2-(pyrid...)
Affinity DataIC50: 31nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9537BDBM9537(N-(4-tert-butylphenyl)-5-{2-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 43nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9544BDBM9544(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 44nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9538BDBM9538(N-[4-(propan-2-yl)phenyl]-5-{2-[2-(pyridin-4-yl)et...)
Affinity DataIC50: 51nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9545BDBM9545(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 58nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9523BDBM9523(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[3-(tr...)
Affinity DataIC50: 64nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9560BDBM9560(N-(3,4-dimethoxyphenyl)-5-{2-[2-(pyridin-4-yl)ethy...)
Affinity DataIC50: 67nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9552BDBM9552(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[3-(tr...)
Affinity DataIC50: 69nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9559BDBM9559(N-(3,4-dichlorophenyl)-5-{2-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 79nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9562BDBM9562(N-(2H-1,3-benzodioxol-5-ylmethyl)-5-{2-[2-(pyridin...)
Affinity DataIC50: 85nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9561BDBM9561(N-[4-methyl-3-(trifluoromethyl)phenyl]-5-{2-[2-(py...)
Affinity DataIC50: 87nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9561BDBM9561(N-[4-methyl-3-(trifluoromethyl)phenyl]-5-{2-[2-(py...)
Affinity DataIC50: 120nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9562BDBM9562(N-(2H-1,3-benzodioxol-5-ylmethyl)-5-{2-[2-(pyridin...)
Affinity DataIC50: 140nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9556BDBM9556(N-(3-methoxyphenyl)-5-{2-[2-(pyridin-4-yl)ethyl]py...)
Affinity DataIC50: 170nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9560BDBM9560(N-(3,4-dimethoxyphenyl)-5-{2-[2-(pyridin-4-yl)ethy...)
Affinity DataIC50: 180nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9539BDBM9539(N-(4-tert-butylphenyl)-5-{3-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 190nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9546BDBM9546(N-[4-(chlorodifluoromethoxy)phenyl]-5-{3-[2-(pyrid...)
Affinity DataIC50: 220nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9523BDBM9523(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[3-(tr...)
Affinity DataIC50: 220nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9539BDBM9539(N-(4-tert-butylphenyl)-5-{3-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 220nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9540BDBM9540(N-[4-(propan-2-yl)phenyl]-5-{3-[2-(pyridin-4-yl)et...)
Affinity DataIC50: 250nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9552BDBM9552(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[3-(tr...)
Affinity DataIC50: 260nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9540BDBM9540(N-[4-(propan-2-yl)phenyl]-5-{3-[2-(pyridin-4-yl)et...)
Affinity DataIC50: 270nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9559BDBM9559(N-(3,4-dichlorophenyl)-5-{2-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 270nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9548BDBM9548(5-{3-[2-(pyridin-4-yl)ethyl]pyridin-4-yl}-N-[4-(tr...)
Affinity DataIC50: 290nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9541BDBM9541(N-(4-tert-butylphenyl)-5-{4-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 310nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9545BDBM9545(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 320nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9547BDBM9547(5-{3-[2-(pyridin-4-yl)ethyl]pyridin-4-yl}-N-[4-(tr...)
Affinity DataIC50: 350nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9550BDBM9550(5-{4-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 360nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9535BDBM9535(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-(quino...)
Affinity DataIC50: 380nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9535BDBM9535(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-(quino...)
Affinity DataIC50: 440nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9549BDBM9549(N-[4-(chlorodifluoromethoxy)phenyl]-5-{4-[2-(pyrid...)
Affinity DataIC50: 440nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9551BDBM9551(5-{4-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 440nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9550BDBM9550(5-{4-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 470nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9553BDBM9553(5-{3-[2-(pyridin-4-yl)ethyl]pyridin-4-yl}-N-[3-(tr...)
Affinity DataIC50: 470nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9541BDBM9541(N-(4-tert-butylphenyl)-5-{4-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 480nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9556BDBM9556(N-(3-methoxyphenyl)-5-{2-[2-(pyridin-4-yl)ethyl]py...)
Affinity DataIC50: 500nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9549BDBM9549(N-[4-(chlorodifluoromethoxy)phenyl]-5-{4-[2-(pyrid...)
Affinity DataIC50: 530nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9554BDBM9554(5-{4-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[3-(tr...)
Affinity DataIC50: 550nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9544BDBM9544(5-{2-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 560nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9524BDBM9524(5-{3-[2-(pyridin-4-yl)ethyl]pyridin-4-yl}-N-[3-(tr...)
Affinity DataIC50: 560nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9538BDBM9538(N-[4-(propan-2-yl)phenyl]-5-{2-[2-(pyridin-4-yl)et...)
Affinity DataIC50: 620nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9551BDBM9551(5-{4-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[4-(tr...)
Affinity DataIC50: 670nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9553BDBM9553(5-{3-[2-(pyridin-4-yl)ethyl]pyridin-4-yl}-N-[3-(tr...)
Affinity DataIC50: 710nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9525BDBM9525(5-{4-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[3-(tr...)
Affinity DataIC50: 720nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9543BDBM9543(N-[4-(chlorodifluoromethoxy)phenyl]-5-{2-[2-(pyrid...)
Affinity DataIC50: 730nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9554BDBM9554(5-{4-[2-(pyridin-4-yl)ethyl]pyridin-3-yl}-N-[3-(tr...)
Affinity DataIC50: 740nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9524BDBM9524(5-{3-[2-(pyridin-4-yl)ethyl]pyridin-4-yl}-N-[3-(tr...)
Affinity DataIC50: 760nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9537BDBM9537(N-(4-tert-butylphenyl)-5-{2-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 770nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9555BDBM9555(N-(3-methylphenyl)-5-{2-[2-(pyridin-4-yl)ethyl]pyr...)
Affinity DataIC50: 770nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandChemical structure of BindingDB Monomer ID 9546BDBM9546(N-[4-(chlorodifluoromethoxy)phenyl]-5-{3-[2-(pyrid...)
Affinity DataIC50: 810nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2006
Entry Details Article
PubMed
Displayed 1 to 50 (of 82 total ) | Next | Last >>
Jump to: