Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50017468
TargetVitamin D3 receptor(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50182484((1R,3R)-5-{2-[1-((1R,5S)-5-adamantan-1-yl-5-hydrox...)
Affinity DataIC50:  50nMAssay Description:Antagonistic activity against human VDR in presence of 1,25(OH)2D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50182485((S)-5-((R)-2-(4-(2-((3R,5R)-3,5-dihydroxy-4-methyl...)
Affinity DataIC50:  300nMAssay Description:Inhibition of transactivation of human VDR in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50182484((1R,3R)-5-{2-[1-((1R,5S)-5-adamantan-1-yl-5-hydrox...)
Affinity DataIC50:  400nMAssay Description:Inhibition of transactivation of human VDR in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed