Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50037675
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50117108(4-[3-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataKi:  0.0140nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50117109(1-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]...)
Affinity DataKi:  0.0460nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183515(CHEMBL383714 | CHEMBL534936 | 5-[[(2-pyridyl)amino...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183525(CHEMBL203797 | CHEMBL534489 | 5-[[(3-pyridyl)amino...)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183515(CHEMBL383714 | CHEMBL534936 | 5-[[(2-pyridyl)amino...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183525(CHEMBL203797 | CHEMBL534489 | 5-[[(3-pyridyl)amino...)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183526(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183530(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183522(5-[[(2-methyl-thiophen-3-yl)amino]carbonyl]amino-8...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183520(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183528(5-[[(5-methyl-thiophen-2-yl)amino]carbonyl]amino-8...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183527(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183516(5-[[(3-furyl)amino]carbonyl]amino-8-methyl-2-(2-fu...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183529(5-[[(benzofuran-2-yl)amino]carbonyl]amino-8-methyl...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183524(5-[[(2-furyl)amino]carbonyl]amino-8-methyl-2-(2-fu...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183523(4-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183521(4-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183520(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183529(5-[[(benzofuran-2-yl)amino]carbonyl]amino-8-methyl...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183526(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50117109(1-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183527(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50117108(4-[3-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183530(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183519(5-[[(quinolin-2-yl)amino]carbonyl]amino-8-methyl-2...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183525(CHEMBL203797 | CHEMBL534489 | 5-[[(3-pyridyl)amino...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183515(CHEMBL383714 | CHEMBL534936 | 5-[[(2-pyridyl)amino...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183523(4-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183525(CHEMBL203797 | CHEMBL534489 | 5-[[(3-pyridyl)amino...)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183515(CHEMBL383714 | CHEMBL534936 | 5-[[(2-pyridyl)amino...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183515(CHEMBL383714 | CHEMBL534936 | 5-[[(2-pyridyl)amino...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183525(CHEMBL203797 | CHEMBL534489 | 5-[[(3-pyridyl)amino...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183520(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 244nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183525(CHEMBL203797 | CHEMBL534489 | 5-[[(3-pyridyl)amino...)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183529(5-[[(benzofuran-2-yl)amino]carbonyl]amino-8-methyl...)
Affinity DataIC50: 250nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50117109(1-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183527(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 260nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183515(CHEMBL383714 | CHEMBL534936 | 5-[[(2-pyridyl)amino...)
Affinity DataKi:  265nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183526(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 280nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183521(4-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  282nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183530(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 320nMAssay Description:Inhibition of NECA-stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183520(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183524(5-[[(2-furyl)amino]carbonyl]amino-8-methyl-2-(2-fu...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50117108(4-[3-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2...)
Affinity DataKi:  355nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183526(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183516(5-[[(3-furyl)amino]carbonyl]amino-8-methyl-2-(2-fu...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183522(5-[[(2-methyl-thiophen-3-yl)amino]carbonyl]amino-8...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183527(3-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183530(2-[3-(2-furan-2-yl-8-methy-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50183519(5-[[(quinolin-2-yl)amino]carbonyl]amino-8-methyl-2...)
Affinity DataKi:  810nMAssay Description:Displacement of [3H]ZM-241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 72 total ) | Next | Last >>
Jump to: