Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50017712
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185537(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185556(2-(2-(3-(4-(trifluoromethyl)phenethyl)-1,2,4-oxadi...)
Affinity DataIC50:  49nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185547(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50:  58nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185544(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50:  62nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185568((2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-1H...)
Affinity DataIC50:  62nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185571(2-(2-(3-(3-cyclohexylpropyl)-1,2,4-oxadiazol-5-yl)...)
Affinity DataIC50:  71nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185541(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50:  95nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185554(2-(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-y...)
Affinity DataIC50:  97nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185574(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50:  120nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185538(2-(2-(3-(2-cyclohexylethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185537(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50:  199nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185562(3-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50:  210nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185547(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50:  223nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185578(CHEMBL211310 | dimethyl-(2-{2-[3-(2-p-tolyl-ethyl)...)
Affinity DataIC50:  230nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185568((2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-1H...)
Affinity DataIC50:  233nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185571(2-(2-(3-(3-cyclohexylpropyl)-1,2,4-oxadiazol-5-yl)...)
Affinity DataIC50:  294nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185576(2-(2-(3-((4-chlorophenoxy)methyl)-1,2,4-oxadiazol-...)
Affinity DataIC50:  410nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185556(2-(2-(3-(4-(trifluoromethyl)phenethyl)-1,2,4-oxadi...)
Affinity DataIC50:  421nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185577(2-(2-(3-(2-(bicyclo[2.2.1]heptan-2-yl)ethyl)-1,2,4...)
Affinity DataIC50:  440nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185552(2-(2-(3-(cyclohexylmethyl)-1,2,4-oxadiazol-5-yl)-1...)
Affinity DataIC50:  440nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185554(2-(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-y...)
Affinity DataIC50:  450nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185582(2-(2-(3-(4-chlorobenzyl)-1,2,4-oxadiazol-5-yl)-1H-...)
Affinity DataIC50:  450nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185549(2-(2-(3-(4-fluorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50:  450nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185567(2-(2-(3-(4-methoxyphenethyl)-1,2,4-oxadiazol-5-yl)...)
Affinity DataIC50:  560nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185575(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50:  568nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185545(2-(2-(3-(2-cyclopentylethyl)-1,2,4-oxadiazol-5-yl)...)
Affinity DataIC50:  580nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185553(2-(2-(5-(4-chlorophenethyl)-1,2,4-oxadiazol-3-yl)-...)
Affinity DataIC50:  600nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185541(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50:  632nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185544(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50:  899nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185580(2-(2-(3-(3,3-dimethylbutyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185579(4-(2-(5-(4-(2-(dimethylamino)ethyl)-1H-indol-2-yl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185572(CHEMBL378513 | N-(3-(4-chlorophenyl)propyl)-4-(2-(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185570(2-(2-(3-isopentyl-1,2,4-oxadiazol-5-yl)-1H-indol-4...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185573(CHEMBL209051 | N,N-dimethyl-2-(2-(3-(2-(pyridin-4-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185566(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185569(CHEMBL377358 | N,N-dimethyl-2-(2-(3-(3-(pyrrolidin...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185563(CHEMBL209507 | N,N-dimethyl-2-(2-(3-(2-(tetrahydro...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185564(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4,5...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185561(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185565(2-(2-(3-(3-methoxy-3-methylbutyl)-1,2,4-oxadiazol-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185581(CHEMBL377161 | N,N-dimethyl-2-(2-(3-(2-(pyridin-3-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185558(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185560(2-(2-(3-butyl-1,2,4-oxadiazol-5-yl)-1H-indol-4-yl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185557(CHEMBL210043 | N-(4-chlorophenethyl)-4-(2-(dimethy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185555(2-(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185551(CHEMBL377228 | N,N-dimethyl-2-(2-(3-(2-(pyridin-2-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185550(CHEMBL377021 | N,N-dimethyl-2-(2-(3-phenethyl-1,2,...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185548(CHEMBL211234 | N,N-dimethyl-2-(2-(3-propyl-1,2,4-o...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185546(2-(2-(5-(4-chlorophenethyl)-1,3,4-oxadiazol-2-yl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185543(2-(2-(3-(3-(4-chlorophenyl)propyl)-1,2,4-oxadiazol...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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