Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50017815
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187004BDBM50187004(3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187007BDBM50187007(5-chloro-3-(3,4-dioxo-2-(phenylamino)cyclobut-1-en...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187002BDBM50187002(CHEMBL209859 | 4-(3,4-dioxo-2-(phenylamino)cyclobu...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187003BDBM50187003(CHEMBL214047 | CHEMBL218964 | 3-(3,4-dioxo-2-(pent...)
Affinity DataIC50: 5nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186997BDBM50186997(3-(2-(cyclopentylamino)-3,4-dioxocyclobut-1-enylam...)
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187016BDBM50187016(2-hydroxy-3-(2-(isopropylamino)-3,4-dioxocyclobut-...)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187015BDBM50187015(3-(2-(cyclohexylamino)-3,4-dioxocyclobut-1-enylami...)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187014BDBM50187014(3-(2-(tert-butylamino)-3,4-dioxocyclobut-1-enylami...)
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187010BDBM50187010(3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187011BDBM50187011(3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187001BDBM50187001(CHEMBL379438 | 3-(2-hydroxy-4-nitrophenylamino)-4-...)
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186999BDBM50186999(3-(2-(furan-2-ylmethylamino)-3,4-dioxocyclobut-1-e...)
Affinity DataIC50: 41nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187017BDBM50187017(methyl 3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enyl...)
Affinity DataIC50: 53nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186998BDBM50186998(3-(2-hydroxy-5-nitrophenylamino)-4-(phenylamino)cy...)
Affinity DataIC50: 56nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187019BDBM50187019(3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50: 65nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187009BDBM50187009(3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50: 74nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187012BDBM50187012(N-benzyl-3-(3,4-dioxo-2-(phenylamino)cyclobut-1-en...)
Affinity DataIC50: 139nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187020BDBM50187020(3-(3,4-dioxo-2-(tetrahydro-2H-pyran-4-ylamino)cycl...)
Affinity DataIC50: 171nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187006BDBM50187006(CHEMBL424694 | 3-(2-hydroxyphenylamino)-4-(phenyla...)
Affinity DataIC50: 476nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187008BDBM50187008((R)-3-(2-(2,3-dihydro-1H-inden-1-ylamino)-3,4-diox...)
Affinity DataIC50: 548nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187021BDBM50187021(3-(3,4-dioxo-2-(phenethylamino)cyclobut-1-enylamin...)
Affinity DataIC50: 926nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187000BDBM50187000(3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187013BDBM50187013(4-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50: 3.10E+3nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187018BDBM50187018(2-hydroxy-N,N-dimethyl-3-(2-(methyl(phenyl)amino)-...)
Affinity DataIC50: 7.20E+3nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187005BDBM50187005(3-(4-nitrophenylamino)-4-(phenylamino)cyclobut-3-e...)
Affinity DataIC50: 8.60E+3nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187022BDBM50187022(3-((2-hydroxyphenyl)(methyl)amino)-4-(phenylamino)...)
Affinity DataIC50: 2.86E+4nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed