Compile Data Set for Download or QSAR
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Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50017925
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188476(CHEMBL209876 | N-4-[4-(3-chloro-2-methoxyphenyl)pi...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188474(CHEMBL426863 | N-[4-[4-(2,3-difluorophenyl)piperaz...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188478(CHEMBL210461 | N-[4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]spiperone from human D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from human D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from human D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]spiperone from human D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188477(CHEMBL208847 | N-4-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188474(CHEMBL426863 | N-[4-[4-(2,3-difluorophenyl)piperaz...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188476(CHEMBL209876 | N-4-[4-(3-chloro-2-methoxyphenyl)pi...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188476(CHEMBL209876 | N-4-[4-(3-chloro-2-methoxyphenyl)pi...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]spiperone from human D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188476(CHEMBL209876 | N-4-[4-(3-chloro-2-methoxyphenyl)pi...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188474(CHEMBL426863 | N-[4-[4-(2,3-difluorophenyl)piperaz...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]spiperone from human D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188476(CHEMBL209876 | N-4-[4-(3-chloro-2-methoxyphenyl)pi...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]spiperone from human D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188477(CHEMBL208847 | N-4-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]spiperone from human D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188474(CHEMBL426863 | N-[4-[4-(2,3-difluorophenyl)piperaz...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188478(CHEMBL210461 | N-[4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188478(CHEMBL210461 | N-[4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]spiperone from human D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188477(CHEMBL208847 | N-4-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188477(CHEMBL208847 | N-4-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]spiperone from human D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188477(CHEMBL208847 | N-4-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]spiperone from human D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188478(CHEMBL210461 | N-[4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]spiperone from human D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]spiperone from human D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188474(CHEMBL426863 | N-[4-[4-(2,3-difluorophenyl)piperaz...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]SCH 23390 from D1 receptor of porcine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188474(CHEMBL426863 | N-[4-[4-(2,3-difluorophenyl)piperaz...)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]SCH 23390 from D1 receptor of porcine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188478(CHEMBL210461 | N-[4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  660nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188475((R)-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]...)
Affinity DataKi:  660nMAssay Description:Displacement of [3H]SCH 23390 from D1 receptor of porcine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  760nMAssay Description:Displacement of [3H]SCH 23390 from D1 receptor of porcine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188477(CHEMBL208847 | N-4-(4-(2-methoxyphenyl)piperazin-1...)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]SCH 23390 from D1 receptor of porcine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188476(CHEMBL209876 | N-4-[4-(3-chloro-2-methoxyphenyl)pi...)
Affinity DataKi:  970nMAssay Description:Displacement of [3H]SCH 23390 from D1 receptor of porcine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(1A) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188478(CHEMBL210461 | N-[4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]SCH 23390 from D1 receptor of porcine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataEC50:  1.80nMAssay Description:Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as rate of [3H]thymidine incorporation by mitogenesis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataEC50:  2.60nMAssay Description:Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as rate of [3H]thymidine incorporation by mitogenesis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188478(CHEMBL210461 | N-[4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataEC50:  110nMAssay Description:Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as rate of [3H]thymidine incorporation by mitogenesis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50188476(CHEMBL209876 | N-4-[4-(3-chloro-2-methoxyphenyl)pi...)
Affinity DataEC50:  18nMAssay Description:Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as rate of [3H]thymidine incorporation by mitogenesis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed