Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50017998 Sort by
TargetLutropin-choriogonadotropic hormone receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189775(N-tert-butyl-5-amino-4-(2,3-dimethoxyphenyl)-2-(me...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189776(tert-butyl 5-amino-4-(3-methoxyphenyl)-2-(methylth...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189773(N-tert-butyl-5-amino-4-(2-fluoro-3-methoxyphenyl)-...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189777(N-tert-butyl-5-amino-4-(3-fluorophenyl)-2-(methylt...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189774(N-tert-butyl-5-amino-4-(3-hydroxyphenyl)-2-(methyl...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189778(cid_9887381 | N-tert-butyl-5-amino-4-(3-methoxyphe...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189779(N-tert-butyl-5-amino-4-(3-methoxyphenyl)-N-methyl-...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThyrotropin receptor(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50189778(cid_9887381 | N-tert-butyl-5-amino-4-(3-methoxyphe...)
Affinity DataEC50:  6.50E+3nMAssay Description:Agonist activity at TSHR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed