TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity against human TRPV1 assessed as inhibition of acid-induced calcium influx by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 2C19More data for this Ligand-Target Pair
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 2D6More data for this Ligand-Target Pair
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 2C9More data for this Ligand-Target Pair
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 1A2More data for this Ligand-Target Pair
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 3A4More data for this Ligand-Target Pair