Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50018022
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50189987(6-phenyl-N-(quinolin-7-yl)nicotinamide | CHEMBL213...)
Affinity DataIC50:  7.90nMAssay Description:Antagonist activity against human TRPV1 assessed as inhibition of acid-induced calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50189987(6-phenyl-N-(quinolin-7-yl)nicotinamide | CHEMBL213...)
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50189987(6-phenyl-N-(quinolin-7-yl)nicotinamide | CHEMBL213...)
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50189987(6-phenyl-N-(quinolin-7-yl)nicotinamide | CHEMBL213...)
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50189987(6-phenyl-N-(quinolin-7-yl)nicotinamide | CHEMBL213...)
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50189987(6-phenyl-N-(quinolin-7-yl)nicotinamide | CHEMBL213...)
Affinity DataIC50: >1.80E+4nMAssay Description:Inhibition of cytochrome P450 3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed