Compile Data Set for Download or QSAR
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Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 5775
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM50261631(3-(3-(trifluoromethyl)benzylthio)-5-sec-butyl-4-hy...)
Affinity DataIC50:  6.00E+4nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93272(Tetramic acid, 72)
Affinity DataIC50:  1.05E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93271(Tetramic acid, 56)
Affinity DataIC50:  1.45E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93267(Tetramic acid, 25)
Affinity DataIC50:  1.94E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93270(Tetramic acid, 44)
Affinity DataIC50: >2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93269(Tetramic acid, 43)
Affinity DataIC50:  2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93268(Tetramic acid, 30)
Affinity DataIC50:  2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93277(N-Substituted tetramic acid, 91)
Affinity DataIC50: >2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93276(N-Substituted tetramic acid, 89)
Affinity DataIC50: >2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93275(Tetramic acid, 77)
Affinity DataIC50: >2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93274(Tetramic acid, 76)
Affinity DataIC50: >2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93273(Tetramic acid, 74)
Affinity DataIC50: >2.00E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93278(N-Substituted tetramic acid, 92)
Affinity DataIC50:  2.12E+5nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93286(N-Substituted tetramic acid, 100)
Affinity DataIC50:  1.39E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93279(N-Substituted tetramic acid, 93)
Affinity DataIC50:  1.84E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93289(N-Substituted tetramic acid, 101)
Affinity DataIC50: >2.00E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93287(Sulfo-tetramic acid, 108)
Affinity DataIC50: >2.00E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93288(Sulfo-tetramic acid, 109)
Affinity DataIC50: >2.00E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93285(N-Substituted tetramic acid, 99)
Affinity DataIC50:  2.12E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93282(N-Substituted tetramic acid, 96)
Affinity DataIC50:  2.41E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93280(N-Substituted tetramic acid, 94)
Affinity DataIC50:  2.58E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93281(N-Substituted tetramic acid, 95)
Affinity DataIC50:  2.65E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93284(N-Substituted tetramic acid, 98)
Affinity DataIC50:  4.24E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandPNGBDBM93283(N-Substituted tetramic acid, 97)
Affinity DataIC50:  4.59E+8nMT: 20°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed