Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50018158
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192093(cis-5-(4-chlorobenzyl)-N-benzyl-6-oxomorpholine-3-...)
Affinity DataIC50: 450nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192090(cis-5-isopropyl-6-oxo-morpholine-3-carboxylic acid...)
Affinity DataIC50: 990nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192085(cis-N,5-dibenzyl-6-oxomorpholine-3-carboxamide | C...)
Affinity DataIC50: 1.01E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192088(cis-5-(4-nitrobenzyl)-N-benzyl-6-oxomorpholine-3-c...)
Affinity DataIC50: 1.13E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192092(cis-N-benzyl-5-((R)-sec-butyl)-6-oxomorpholine-3-c...)
Affinity DataIC50: 1.22E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192089(trans-5-(4-chlorobenzyl)-6-oxo-N-((S)-1-phenylethy...)
Affinity DataIC50: 1.33E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50117922(CHEMBL45816 | Methoxy-acetic acid 2-(2-{[3-(1H-ben...)
Affinity DataIC50: 1.34E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192086(cis-5-(4-hydroxybenzyl)-6-oxo-N-((S)-1-phenylethyl...)
Affinity DataIC50: 1.39E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192087(trans-5-(4-fluorobenzyl)-6-oxo-N-((S)-1-phenylethy...)
Affinity DataIC50: 1.48E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192097(cis-5-(4-chlorobenzyl)-6-oxo-N-((S)-1-phenylethyl)...)
Affinity DataIC50: 1.61E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192096(cis-N-benzyl-5-(2-(methylthio)ethyl)-6-oxomorpholi...)
Affinity DataIC50: 1.86E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192094(cis-5-(4-methoxybenzyl)-N-benzyl-6-oxomorpholine-3...)
Affinity DataIC50: 2.04E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192095(cis-5-(4-nitrobenzyl)-6-oxo-N-((S)-1-phenylethyl)m...)
Affinity DataIC50: 2.13E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192091(cis-5-benzyl-N-cyclohexyl-6-oxomorpholine-3-carbox...)
Affinity DataIC50: 2.18E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50192084(cis-5-(4-fluorobenzyl)-N-benzyl-6-oxomorpholine-3-...)
Affinity DataIC50: 2.75E+3nMAssay Description:Ability to block calcium channel T type 3.1v expressed in HEK293 cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed