Compile Data Set for Download or QSAR
Report error Found 129 Enz. Inhib. hit(s) with all data for entry = 50018474
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196109((2,3-dimethylquinolin-4-yl)-[4-(octahydro-2H-pyrid...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196123({2-methyl-4-[4-(3,3,4-trimethylpiperazin-1-yl)phen...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196117(1-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-2...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196142([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2-methyl-3...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196132([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,8-te...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196139((3-methylquinolin-4-yl)-[4-(3,3,4-trimethylpiperaz...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196107({7-chloro-4-[4-(3,3,4-trimethylpiperazin-1-yl)phen...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196118({4-[4-(3,3,4-trimethylpiperazin-1-yl)phenylamino]q...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196146([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,8-trim...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196129({4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-2-m...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196145((R)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196125((R)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7-...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50418050(CHEMBL1689423)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196131([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(3-methylqu...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196147((3-ethyl-2,8-dimethylquinolin-4-yl)-[4-(4-methyl-[...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196126((R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196116((R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196113([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7-trim...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196120([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(6-fluoro-2...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196136((3-ethyl-2-methylquinolin-4-yl)-[4-(4-methylpipera...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196135(TCMDC-123912 | Acridin-9-yl-[4-(4-methyl-piperazin...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196128((3-benzyl-2-methylquinolin-4-yl)-[4-(4-methylpiper...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196141((2,3-dimethylquinolin-4-yl)-[4-(4-methylpiperazin-...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196130((2-methyl-3-phenylquinolin-4-yl)-[4-(4-methylpiper...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196122(N-(4-(4-ethylpiperazin-1-yl)phenyl)acridin-9-amine...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196127((R)-{4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196115({4-[4-(3,4-dimethylpiperazin-1-yl)phenylamino]-6-f...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196108({6-fluoro-4-[4-(3,3,4-trimethylpiperazin-1-yl)phen...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196119((3-isopropyl-2-methylquinolin-4-yl)-[4-(4-methylpi...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196140((S)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7-...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196106(N-(2-diethylaminoethyl)-N'-(3-ethyl-2,8-dimethylqu...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196124((S)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196121([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5-trim...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196128((3-benzyl-2-methylquinolin-4-yl)-[4-(4-methylpiper...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2B expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196114(N-(2,3-dimethylquinolin-4-yl)-N'-(2-pyrrolidin-1-y...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196143(4-(3,4-dimethylpiperazin-1-yl)phenyl]-(3-ethyl-2-m...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196148([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5,7-te...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196138((5-chloro-2,3-dimethylquinolin-4-yl)-[4-(3,4-dimet...)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196134((R)-{4-[4-(3-methylpiperazin-1-yl)phenylamino]quin...)
Affinity DataKi:  205nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196112([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5,8-te...)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196107({7-chloro-4-[4-(3,3,4-trimethylpiperazin-1-yl)phen...)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2B expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196137([4-(4-methylpiperazin-1-yl)phenyl]-(2-methylquinol...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2A expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196128((3-benzyl-2-methylquinolin-4-yl)-[4-(4-methylpiper...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2A expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196132([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,8-te...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2B expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196145((R)-[4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,7,...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2B expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196143(4-(3,4-dimethylpiperazin-1-yl)phenyl]-(3-ethyl-2-m...)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2A expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196148([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5,7-te...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2A expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196121([4-(3,4-dimethylpiperazin-1-yl)phenyl]-(2,3,5-trim...)
Affinity DataKi:  680nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2A expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196137([4-(4-methylpiperazin-1-yl)phenyl]-(2-methylquinol...)
Affinity DataKi:  690nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196109((2,3-dimethylquinolin-4-yl)-[4-(octahydro-2H-pyrid...)
Affinity DataKi:  715nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2A expressed in S115 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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