Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50038434
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376416(CHEMBL253952)
Affinity DataIC50:  99nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50150998(((4-Methoxy-phenoxycarbonyl)-{4-[2-(5-methyl-2-phe...)
Affinity DataIC50:  188nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50150998(((4-Methoxy-phenoxycarbonyl)-{4-[2-(5-methyl-2-phe...)
Affinity DataIC50:  247nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50150998(((4-Methoxy-phenoxycarbonyl)-{4-[2-(5-methyl-2-phe...)
Affinity DataIC50:  1.41E+3nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376416(CHEMBL253952)
Affinity DataIC50:  2.05E+3nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376415(CHEMBL429671)
Affinity DataIC50:  3.09E+3nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376414(CHEMBL254989)
Affinity DataIC50:  3.74E+3nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376412(CHEMBL254347)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376413(CHEMBL444373)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376415(CHEMBL429671)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376414(CHEMBL254989)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376411(CHEMBL401829)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376413(CHEMBL444373)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376412(CHEMBL254347)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376411(CHEMBL401829)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376410(CHEMBL257761)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376410(CHEMBL257761)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity at PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376416(CHEMBL253952)
Affinity DataIC50:  1.98E+4nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376413(CHEMBL444373)
Affinity DataIC50: >2.00E+4nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376412(CHEMBL254347)
Affinity DataIC50: >2.50E+4nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376411(CHEMBL401829)
Affinity DataIC50: >2.50E+4nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376410(CHEMBL257761)
Affinity DataIC50: >2.50E+4nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376414(CHEMBL254989)
Affinity DataIC50: >2.50E+4nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376415(CHEMBL429671)
Affinity DataIC50: >2.50E+4nMAssay Description:Agonist activity at PPAR gamma in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376414(CHEMBL254989)
Affinity DataEC50:  6.89E+3nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376413(CHEMBL444373)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376410(CHEMBL257761)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376411(CHEMBL401829)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50150998(((4-Methoxy-phenoxycarbonyl)-{4-[2-(5-methyl-2-phe...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376416(CHEMBL253952)
Affinity DataEC50:  260nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376412(CHEMBL254347)
Affinity DataEC50:  1.81E+4nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50376415(CHEMBL429671)
Affinity DataEC50:  1.94E+3nMAssay Description:Agonist activity at PPAR alpha in human HEK cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed