Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50018841
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199575BDBM50199575((1-(4-chlorophenoxy)-9-((1-methylpiperidin-4-yl)me...)
Affinity DataIC50: 11nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199586BDBM50199586(2-(4-((1-(4-chlorophenoxy)-3-(1-methylpiperazine-4...)
Affinity DataIC50: 14nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199587BDBM50199587((1-(4-chlorophenoxy)-9-(piperidin-4-ylmethyl)-9H-c...)
Affinity DataIC50: 16nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199580BDBM50199580((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoro-1-methyl...)
Affinity DataIC50: 28nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199584BDBM50199584((1-(4-chlorophenoxy)-9-((3-fluoro-1,2,5,6-tetrahyd...)
Affinity DataIC50: 43nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199577BDBM50199577((1-(4-chlorophenoxy)-9-(3-(piperidin-1-yl)propyl)-...)
Affinity DataIC50: 50nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199579BDBM50199579(1-(4-chlorophenoxy)-N-(2-(dimethylamino)ethyl)-9-(...)
Affinity DataIC50: 50nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199585BDBM50199585((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50: 51nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199570BDBM50199570((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin...)
Affinity DataIC50: 53nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199574BDBM50199574((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoro-1-methyl...)
Affinity DataIC50: 95nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199573BDBM50199573((1-(4-chlorophenoxy)-9-(piperidin-3-ylmethyl)-9H-c...)
Affinity DataIC50: 107nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199581BDBM50199581((1-(4-chlorophenoxy)-9-(((3R,4S)-1-cyclopropyl-3-f...)
Affinity DataIC50: 186nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199572BDBM50199572(1-(4-chlorophenoxy)-N-(2-(dimethylamino)ethyl)-9-(...)
Affinity DataIC50: 191nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199571BDBM50199571(1-(4-chlorophenoxy)-N-((1-ethylpyrrolidin-2-yl)met...)
Affinity DataIC50: 263nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199583BDBM50199583((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin...)
Affinity DataIC50: 467nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199588BDBM50199588((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50: 832nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199589BDBM50199589((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin...)
Affinity DataIC50: 871nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199590BDBM50199590(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-...)
Affinity DataIC50: 1.86E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199578BDBM50199578((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50: 1.91E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199582BDBM50199582((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50: 2.88E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199591BDBM50199591((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50: 7.76E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199576BDBM50199576((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50: 9.77E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50199569BDBM50199569(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-...)
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed