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Found 27 Enz. Inhib. hit(s) with all data for entry = 50018905
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200200((S)-2-amino-N-hydroxy-3-(4-hydroxyphenyl)propanami...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200197((S)-2-amino-N-hydroxy-3-(4-hydroxyphenyl)propaneth...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200187((S)-2-amino-N-hydroxy-3-(4-iodophenyl)propanamide ...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200208((S)-2-amino-N-hydroxy-3-(4-isopropylphenyl)propana...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200198((S)-2-amino-N-hydroxy-3-(4-hydroxy-3,5-diiodopheny...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200190((S)-2-amino-N-hydroxy-3-(2-iodophenyl)propanamide ...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200189((S)-2-amino-N-hydroxy-3-[4-(nitrophenyl)phenyl]pro...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200196((S)-2-amino-3-(4-bromophenyl)-N-hydroxypropionamid...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200201((S)-2-amino-N-hydroxy-3-[3-(nitrophenyl)phenyl]pro...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200188((S)-2-amino-3-(4-chlorophenyl)-N-hydroxypropanamid...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200206((S)-2-amino-N-hydroxy-3-(4-nitrophenyl)propanamide...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200203((S)-2-amino-N-hydroxy-3-p-tolylpropionamide | CHEM...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200200((S)-2-amino-N-hydroxy-3-(4-hydroxyphenyl)propanami...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200205((S)-2-amino-3-(4-fluorophenyl)-N-hydroxypropanamid...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200184((S)-2-amino-N-hydroxy-3-[4-(phenyl)phenyl]propanam...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200194((S)-2-amino-N-hydroxy-3-phenylpropanamide | CHEMBL...)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200193((S)-2-amino-3-(3,4-difluorophenyl)-N-hydroxypropan...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200185((S)-2-amino-N-hydroxy-4-(4-hydroxyphenyl)butanamid...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200207((S)-2-amino-3-(4-azidophenyl)-N-hydroxypropanamide...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200192((S)-2-amino-3-(4-cyanophenyl)-N-hydroxypropanamide...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200195((S)-2-benzylamino-N-hydroxy-3-(4-hydroxyphenyl)pro...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200202(4-((S)-2-(hydroxycarbamoyl)-2-aminoethyl)phenylbor...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200204((S)-2-amino-3-(4-aminophenyl)-N-hydroxypropanamide...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200186((S)-2-amino-N-hydroxy-2-(4-hydroxyphenyl)acetamide...)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200191((S)-2-amino-3-(4-hydroxyphenyl)propanehydrazide | ...)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200199((S)-N-hydroxy-3-(4-hydroxyphenyl)-2-phenylpropanam...)
Affinity DataIC50:  2.90E+5nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Rhode Island

Curated by ChEMBL
LigandPNGBDBM50200183((S)-2-amino-N-benzyl-N-hydroxy-3-(4-hydroxyphenyl)...)
Affinity DataIC50:  2.91E+5nMAssay Description:Inhibition of CSK measured as poly-E4Y phosphorylation by acid precipitation assay in presence of 0.2 mM CoCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed