Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 2620
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22714(Dihydroxypyrimidine, 5 | N-[(4-fluorophenyl)methyl...)
Affinity DataIC50:  10nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22720(2-[2-(dimethylamino)propan-2-yl]-N-[(4-fluoropheny...)
Affinity DataIC50:  50nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22717(2-benzyl-N-[(4-fluorophenyl)methyl]-5,6-dihydroxyp...)
Affinity DataIC50:  50nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22663(JMC496646 Compound 6 | N-[(4-fluorophenyl)methyl]-...)
Affinity DataIC50:  60nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22715(Dihydroxypyrimidine, 7 | N-[(4-fluorophenyl)methyl...)
Affinity DataIC50:  60nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22628(JMC51861 Compound 4 | N-Me-pyrimidone deriv., 27 |...)
Affinity DataIC50:  60nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22716(Dihydroxypyrimidine, 8 | N-benzyl-5,6-dihydroxy-2-...)
Affinity DataIC50:  70nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22664(2-[1-(dimethylamino)ethyl]-N-[(4-fluorophenyl)meth...)
Affinity DataIC50:  80nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22713(Dihydroxypyrimidine, 4a | N-benzyl-5,6-dihydroxy-2...)
Affinity DataIC50:  85nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22609(JMC496646 Compound 14 | N-[(4-fluorophenyl)methyl]...)
Affinity DataIC50:  200nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22719(2-[(dimethylamino)methyl]-N-[(4-fluorophenyl)methy...)
Affinity DataIC50:  200nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22718(2-[(dimethylamino)(phenyl)methyl]-N-[(4-fluorophen...)
Affinity DataIC50:  200nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Irbm-Mrl

LigandPNGBDBM22611(JMC496646 Compound 16 | N-Me-pyrimidone deriv., 11...)
Affinity DataIC50:  210nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed