Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50025141
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
National Center For Drug Screening

Curated by ChEMBL
LigandPNGBDBM50260245(1,3-bis(4-(cyclopentanecarboxamido)benzamido)-2,4-...)
Affinity DataKi:  287nMAssay Description:Displacement of [125I]GLP1 from rat GLP1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
National Center For Drug Screening

Curated by ChEMBL
LigandPNGBDBM50260246(1,3-bis(4-(tert-butoxycarbonyl)benzamido)-2,4-bis(...)
Affinity DataKi:  1.47E+3nMAssay Description:Displacement of [125I]GLP1 from rat GLP1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
National Center For Drug Screening

Curated by ChEMBL
LigandPNGBDBM50260245(1,3-bis(4-(cyclopentanecarboxamido)benzamido)-2,4-...)
Affinity DataEC50:  1.08E+3nMAssay Description:Agonist activity at rat GLP1 receptor expressed in HEK293 cells assessed as cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
National Center For Drug Screening

Curated by ChEMBL
LigandPNGBDBM50260246(1,3-bis(4-(tert-butoxycarbonyl)benzamido)-2,4-bis(...)
Affinity DataEC50:  2.73E+3nMAssay Description:Agonist activity at rat GLP1 receptor expressed in HEK293 cells assessed as cAMP releaseMore data for this Ligand-Target Pair