Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 2603
LigandChemical structure of BindingDB Monomer ID 22503BDBM22503(2-(4-{[(4-phenylphenyl)methyl]amino}phenyl)cyclopr...)
Affinity DataEC50:  40nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22497BDBM22497(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)cyclop...)
Affinity DataEC50:  50nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22496BDBM22496(CHEMBL207881 | 3-(4-{[(3-phenoxyphenyl)methyl]amin...)
Affinity DataEC50:  79nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22528BDBM22528(3-(4-{[(4-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  195nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22508BDBM22508(3-(4-{[(3,4-dichlorophenyl)methyl]amino}phenyl)pro...)
Affinity DataEC50:  251nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22502BDBM22502(3-(4-{[(4-phenylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  251nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22498BDBM22498(3-(3-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  398nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22504BDBM22504(3-(3-{[(4-phenylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  501nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22509BDBM22509(3-{4-[(naphthalen-2-ylmethyl)amino]phenyl}propanoi...)
Affinity DataEC50:  794nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22510BDBM22510(3-(4-{[(3-bromophenyl)methyl]amino}phenyl)propanoi...)
Affinity DataEC50:  794nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22524BDBM22524(3-(4-{[(4-methoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  1.26E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22505BDBM22505(4-(4-{[(4-phenylphenyl)methyl]amino}phenyl)butanoi...)
Affinity DataEC50:  1.59E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22511BDBM22511(3-(4-{[(5-chlorothiophen-2-yl)methyl]amino}phenyl)...)
Affinity DataEC50:  2.00E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22512BDBM22512(3-[4-({[4-(trifluoromethyl)phenyl]methyl}amino)phe...)
Affinity DataEC50:  2.00E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22499BDBM22499(4-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)butano...)
Affinity DataEC50:  3.16E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22513BDBM22513(3-(4-{[(2-chlorophenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  3.98E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22514BDBM22514(3-(4-{[(4-methylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  3.98E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22501BDBM22501(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)acetic...)
Affinity DataEC50:  3.98E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22515BDBM22515(3-(4-{[(3-fluorophenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  5.01E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22516BDBM22516(3-[4-({[2-chloro-5-(trifluoromethyl)pyridin-3-yl]m...)
Affinity DataEC50:  5.01E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22517BDBM22517(3-[4-(benzylamino)phenyl]propanoic acid | carboxyl...)
Affinity DataEC50:  7.94E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22507BDBM22507(2-(4-{[(4-phenylphenyl)methyl]amino}phenyl)acetic ...)
Affinity DataEC50:  1.23E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22500BDBM22500(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  1.66E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22525BDBM22525(3-(4-{[(3-carbamoylphenyl)methyl]amino}phenyl)prop...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22526BDBM22526(3-{4-[(1H-imidazol-2-ylmethyl)amino]phenyl}propano...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22527BDBM22527(3-(4-{[(3-methanesulfonamidophenyl)methyl]amino}ph...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22518BDBM22518(3-{4-[(pyridin-3-ylmethyl)amino]phenyl}propanoic a...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22519BDBM22519(3-{4-[({4-[(dimethylamino)methyl]phenyl}methyl)ami...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22520BDBM22520(3-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]phenyl}...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22521BDBM22521(4-({[4-(2-carboxyethyl)phenyl]amino}methyl)benzoic...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22506BDBM22506(2-(4-{[(4-phenylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22522BDBM22522(3-(4-{[(4-hydroxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 22523BDBM22523(3-(4-{[(4-cyanophenyl)methyl]amino}phenyl)propanoi...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2008
Entry Details Article
PubMed