Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50019347
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203781((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203782((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203794((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203811((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203802((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203814((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203813((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203816((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203791((2S)-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203800((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  11.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203794((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  11.3nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203802((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  11.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203779((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  15.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203789((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  16.2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataEC50:  17.3nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203811((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  17.6nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203810((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  21.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203814((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  22.2nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  22.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  22.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203813((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  25nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203779((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  25.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203781((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  29.4nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203780((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  29.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203810((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  30.3nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203787((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  33.4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203782((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  33.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203787((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  39.5nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203799((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  51.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203791((2S)-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1...)
Affinity DataEC50:  69.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203789((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  70.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203797((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203797((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203790((2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-me...)
Affinity DataKi:  82.7nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203788((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  86.7nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203790((2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-me...)
Affinity DataEC50:  87.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203798((2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-me...)
Affinity DataKi:  88.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203800((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  91.7nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203807(LPNYNWNSFGLRF-NH2 | CHEMBL374077)
Affinity DataKi:  94.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203786((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  101nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203816((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  103nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203780((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  108nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203786((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  110nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203799((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataEC50:  110nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203795((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  142nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203817((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  162nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
University of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203788((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  197nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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