Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 101 Enz. Inhib. hit(s) with all data for entry = 445
TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  9nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2606(3-(5-chloro-1-methyl-1H-indol-3-yl)-4-(1-methyl-1H...)
Affinity DataIC50:  110nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2607(3-(1,5-dimethyl-1H-indol-3-yl)-4-(1-methyl-1H-indo...)
Affinity DataIC50:  170nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2590((Arylindolyl)maleimide deriv. 12 | 3-(1H-indol-3-y...)
Affinity DataIC50:  220nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2626(3-(1,7-dimethyl-1H-indol-3-yl)-4-(1-methyl-1H-indo...)
Affinity DataIC50:  280nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2591((Arylindolyl)maleimide deriv. 13 | 3,4-bis(1-methy...)
Affinity DataIC50:  300nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2620(3-(6-amino-1-methyl-1H-indol-3-yl)-4-(1-methyl-1H-...)
Affinity DataIC50:  310nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2594((Arylindolyl)maleimide deriv. 16 | 3-(1-methyl-1H-...)
Affinity DataIC50:  360nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2612(3-(1-methyl-1H-indol-3-yl)-4-[1-methyl-5-(methylsu...)
Affinity DataIC50:  380nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2635(3-(1-methyl-1H-indol-3-yl)-4-[1-methyl-2-(methylsu...)
Affinity DataIC50:  440nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2634(3-(1,2-dimethyl-1H-indol-3-yl)-4-(1-methyl-1H-indo...)
Affinity DataIC50:  470nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2580(K252a | methyl (15R,16S,18S)-16-hydroxy-15-methyl-...)
Affinity DataIC50:  470nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2593((Arylindolyl)maleimide deriv. 15 | 3-(1-methyl-1H-...)
Affinity DataIC50:  480nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2608(3-(5-amino-1-methyl-1H-indol-3-yl)-4-(1-methyl-1H-...)
Affinity DataIC50:  490nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2583(3,4-Bis(3-indolyl)-1H-pyrrole-2,5-dione | 3,4-bis(...)
Affinity DataIC50:  550nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2631(3-(1,4-dimethyl-1H-indol-3-yl)-4-(1-methyl-1H-indo...)
Affinity DataIC50:  590nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2610(3-(5-Methoxy-1-methyl-3-indolyl)-4-(1-methyl-3-ind...)
Affinity DataIC50:  600nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2652((Phenylindolyl)maleimide deriv. 74 | 3-(1-methyl-1...)
Affinity DataIC50:  670nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2597((Arylindolyl)maleimide deriv. 19 | 3-(1-methyl-1H-...)
Affinity DataIC50:  810nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2651((Phenylindolyl)maleimide deriv. 73 | 3-(2-chloroph...)
Affinity DataIC50:  900nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2599((Arylindolyl)maleimide deriv. 21 | 3-(1-benzothiop...)
Affinity DataIC50:  900nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2609(3-(5-Hydroxy-1-methyl-3-indolyl)-4-(1-methyl-3-ind...)
Affinity DataIC50:  920nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2653((Phenylindolyl)maleimide deriv. 75 | 3-(1-methyl-1...)
Affinity DataIC50:  950nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2627(3-(7-Amino-1-methyl-3-indolyl)-4-(1-methyl-3-indol...)
Affinity DataIC50:  1.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2628(3-(7-methoxy-1-methyl-1H-indol-3-yl)-4-(1-methyl-1...)
Affinity DataIC50:  1.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2658((Phenylindolyl)maleimide deriv. 80 | 3-(1-methyl-1...)
Affinity DataIC50:  1.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2642((Phenylindolyl)maleimide deriv. 64 | 3-(1-methyl-1...)
Affinity DataIC50:  1.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2636(3-(2-methanesulfinyl-1-methyl-1H-indol-3-yl)-4-(1-...)
Affinity DataIC50:  1.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2622(3-(1-methyl-1H-indol-3-yl)-4-(1-methyl-6-nitro-1H-...)
Affinity DataIC50:  1.10E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2621(3-(6-methoxy-1-methyl-1H-indol-3-yl)-4-(1-methyl-1...)
Affinity DataIC50:  1.10E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2655((Phenylindolyl)maleimide deriv. 77 | 3-(2,5-dimeth...)
Affinity DataIC50:  1.20E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2592((Arylindolyl)maleimide deriv. 14 | 3-(1-benzyl-1H-...)
Affinity DataIC50:  1.20E+3nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2615(Bisindolylmaleimide deriv. 37 | methyl 1-methyl-3-...)
Affinity DataIC50:  1.40E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2629(3-(1-Methyl-3-indolyl)-4-(1-methyl-7-nitro-3-indol...)
Affinity DataIC50:  1.50E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2619(3-(6-chloro-1-methyl-1H-indol-3-yl)-4-(1-methyl-1H...)
Affinity DataIC50:  1.60E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2648((Phenylindolyl)maleimide deriv. 70 | 3-(1-methyl-1...)
Affinity DataIC50:  1.90E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2643((Phenylindolyl)maleimide deriv. 65 | 3-(3-chloroph...)
Affinity DataIC50:  2.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2633(3-(1-methyl-1H-indol-3-yl)-4-(1-methyl-4-nitro-1H-...)
Affinity DataIC50:  2.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2650((Phenylindolyl)maleimide deriv. 72 | 3-(1-methyl-1...)
Affinity DataIC50:  2.20E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2644((Phenylindolyl)maleimide deriv. 66 | 3-(3-bromophe...)
Affinity DataIC50:  2.20E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2630(3-(7-(Acetylamino)-1-methyl-3-indolyl)-4-(1-methyl...)
Affinity DataIC50:  2.40E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2656((Phenylindolyl)maleimide deriv. 78 | 3-(2,6-dichlo...)
Affinity DataIC50:  2.40E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2654((Phenylindolyl)maleimide deriv. 76 | 3-(2,3-dimeth...)
Affinity DataIC50:  2.40E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2614(3-(1-methyl-1H-indol-3-yl)-4-(1-methyl-5-nitro-1H-...)
Affinity DataIC50:  2.50E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2600((Arylindolyl)maleimide deriv. 22 | 3-(1-benzofuran...)
Affinity DataIC50:  2.60E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2598((Arylindolyl)maleimide deriv. 20 | 3-(1-methyl-1H-...)
Affinity DataIC50:  2.80E+3nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2605((Arylindolyl)maleimide deriv. 27 | 3-(1-methyl-1H-...)
Affinity DataIC50:  2.90E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2596((Arylindolyl)maleimide deriv. 18 | 3-(1H-indol-1-y...)
Affinity DataIC50:  3.00E+3nMpH: 7.5 T: 30°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2613(3-(1-Methyl-3-indolyl)-4-(1-methyl-5-(methylsulfin...)
Affinity DataIC50:  3.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2632(3-(4-methoxy-1-methyl-1H-indol-3-yl)-4-(1-methyl-1...)
Affinity DataIC50:  3.00E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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