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Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50019681
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206658((S)-N-(1-(2-amino-3-(4-hydroxy-2,6-dimethylphenyl)...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206658((S)-N-(1-(2-amino-3-(4-hydroxy-2,6-dimethylphenyl)...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206643(CHEMBL390480 | N-(1-((2S,3R)-2-amino-3-(4-hydroxy-...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206643(CHEMBL390480 | N-(1-((2S,3R)-2-amino-3-(4-hydroxy-...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206659((S)-N-(1-(2-amino-3,3-diphenylpropanoyl)piperidin-...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206648(CHEMBL388899 | N-(1-((2S,3S)-2-amino-3-(4-hydroxy-...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206644(CHEMBL395545 | N-(1-(3-amino-3-(4-chlorophenyl)pro...)
Affinity DataKi:  990nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206651((S)-N-(1-(2-amino-3-(naphthalen-2-yl)propanoyl)pip...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206648(CHEMBL388899 | N-(1-((2S,3S)-2-amino-3-(4-hydroxy-...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206653(CHEMBL389109 | N-(1-(3-(3-bromophenyl)propanoyl)pi...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206644(CHEMBL395545 | N-(1-(3-amino-3-(4-chlorophenyl)pro...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206646((S)-N-(1-(2-amino-2-(2,3-dihydro-1H-inden-2-yl)ace...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206645((S)-N-(1-(2-amino-3-(benzo[b]thiophen-3-yl)propano...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206660(CHEMBL231049 | N-(1-(3-amino-3-p-tolylpropanoyl)pi...)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206660(CHEMBL231049 | N-(1-(3-amino-3-p-tolylpropanoyl)pi...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206651((S)-N-(1-(2-amino-3-(naphthalen-2-yl)propanoyl)pip...)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206649(CHEMBL230311 | N-(1-(3-(3-chloro-4-methoxyphenyl)p...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206655((S)-N-(1-(2-amino-3-phenylpropanoyl)piperidin-4-yl...)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206656((R)-N-(1-(2-amino-2-phenylacetyl)piperidin-4-yl)-N...)
Affinity DataKi:  5.10E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206649(CHEMBL230311 | N-(1-(3-(3-chloro-4-methoxyphenyl)p...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206654((S)-N-(1-(2-amino-2-phenylacetyl)piperidin-4-yl)-N...)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206659((S)-N-(1-(2-amino-3,3-diphenylpropanoyl)piperidin-...)
Affinity DataKi:  6.50E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206652((R)-N-(1-(2-amino-3-(4-chlorophenyl)propanoyl)pipe...)
Affinity DataKi:  6.90E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206655((S)-N-(1-(2-amino-3-phenylpropanoyl)piperidin-4-yl...)
Affinity DataKi:  6.90E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206647((S)-N-(1-(2-amino-3-(4-hydroxyphenyl)propanoyl)pip...)
Affinity DataKi:  7.90E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206657(CHEMBL230310 | N-(1-(3-amino-3-(4-methoxyphenyl)pr...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206650((S)-N-(1-(2-amino-3-(thiazol-4-yl)propanoyl)piperi...)
Affinity DataKi:  9.70E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206657(CHEMBL230310 | N-(1-(3-amino-3-(4-methoxyphenyl)pr...)
Affinity DataKi:  9.70E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206653(CHEMBL389109 | N-(1-(3-(3-bromophenyl)propanoyl)pi...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206645((S)-N-(1-(2-amino-3-(benzo[b]thiophen-3-yl)propano...)
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206646((S)-N-(1-(2-amino-2-(2,3-dihydro-1H-inden-2-yl)ace...)
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206647((S)-N-(1-(2-amino-3-(4-hydroxyphenyl)propanoyl)pip...)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206650((S)-N-(1-(2-amino-3-(thiazol-4-yl)propanoyl)piperi...)
Affinity DataKi:  7.60E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50206643(CHEMBL390480 | N-(1-((2S,3R)-2-amino-3-(4-hydroxy-...)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at mu opioid receptor as inhibition of electrically stimulated guinea pig ileum contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed