Compile Data Set for Download or QSAR
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Report error Found 128 Enz. Inhib. hit(s) with all data for entry = 50019866
TargetSerine-protein kinase ATM(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208517(2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one | C...)
Affinity DataIC50:  13nMAssay Description:Inhibition of ATM kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132373(2-(4-(benzo[b]thiophen-3-yl)phenyl)-6-morpholino-4...)
Affinity DataIC50:  160nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132371(2-Morpholin-4-yl-6-(4-naphthalen-1-yl-phenyl)-thio...)
Affinity DataIC50:  160nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132355(2-(4-Chloro-phenyl)-6-morpholin-4-yl-pyran-4-one |...)
Affinity DataIC50:  180nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132361(2-(4-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...)
Affinity DataIC50:  220nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132368(2-[4-(4-Methyl-naphthalen-1-yl)-phenyl]-6-morpholi...)
Affinity DataIC50:  260nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132365(2-(4-Methoxy-phenyl)-6-morpholin-4-yl-thiopyran-4-...)
Affinity DataIC50:  280nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132363(2-(2-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...)
Affinity DataIC50:  310nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132370(2-(4-Fluoro-phenyl)-6-morpholin-4-yl-pyran-4-one |...)
Affinity DataIC50:  350nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208499(6-(2-fluorophenyl)-2-(4-morpholin-4-yl)pyran-4-one...)
Affinity DataIC50:  390nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208505(2-(1H-indol-5-yl)-6-morpholino-4H-pyran-4-one | CH...)
Affinity DataIC50:  400nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208552(6-(4-chlorophenyl)-4-morpholino-2H-pyran-2-one | C...)
Affinity DataIC50:  470nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132358(2-(4-tert-Butyl-phenyl)-6-morpholin-4-yl-pyran-4-o...)
Affinity DataIC50:  480nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208494(2-(4-(6-morpholino-4-oxo-4H-pyran-2-yl)benzyl)isoi...)
Affinity DataIC50:  500nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208558(6-(4-methoxyphenyl)-4-morpholino-2H-pyran-2-one | ...)
Affinity DataIC50:  530nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132369(2-(4-Chloro-phenyl)-6-morpholin-4-yl-thiopyran-4-o...)
Affinity DataIC50:  530nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132356(2-(3-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...)
Affinity DataIC50:  540nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208507(2-(benzo[b]thiophen-2-yl)-6-morpholino-4H-pyran-4-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132364(2-Morpholin-4-yl-6-phenyl-thiopyran-4-one | 2-morp...)
Affinity DataIC50:  650nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208557(CHEMBL222820 | N-[3'-(6-morpholin-4-yl-4-oxo-4H-th...)
Affinity DataIC50:  680nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132367(2-(4-Bromo-phenyl)-6-morpholin-4-yl-thiopyran-4-on...)
Affinity DataIC50:  680nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132360(2-(3-Fluoro-phenyl)-6-morpholin-4-yl-pyran-4-one |...)
Affinity DataIC50:  690nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132354(2-(3-Bromo-phenyl)-6-morpholin-4-yl-thiopyran-4-on...)
Affinity DataIC50:  700nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208500(2-biphenyl-4-yl-6-morpholin-4-yl-pyran-4-one | CHE...)
Affinity DataIC50:  800nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208493(2-(benzofuran-2-yl)-6-morpholino-4H-pyran-4-one | ...)
Affinity DataIC50:  800nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132357((E)-3-[3'-(6-Morpholin-4-yl-4-oxo-4H-thiopyran-2-y...)
Affinity DataIC50:  840nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208495(2-morpholino-6-(quinolin-8-yl)-4H-pyran-4-one | CH...)
Affinity DataIC50:  900nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208533(2-(4-(benzyloxy)phenyl)-6-morpholino-4H-pyran-4-on...)
Affinity DataIC50:  910nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132362(2-(3'-hydroxy-biphenyl-3-yl)-6-morpholin-4-yl-thio...)
Affinity DataIC50:  920nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208515(CHEMBL222815 | benzyl 4-(6-morpholino-4-oxo-4H-pyr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208521(2-(furan-2-yl)-6-morpholino-4H-pyran-4-one | CHEMB...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208546(2-morpholino-6-(4-(trifluoromethoxy)phenyl)-4H-pyr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208510(6-tert-Butyl-2-morpholin-4-yl-4H-thiopyran-4-one |...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132372(2-(4-tert-Butyl-phenyl)-6-morpholin-4-yl-thiopyran...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208542(CHEMBL223667 | methyl 3-(3-(6-morpholino-4-oxo-4H-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208518(2-morpholino-6-(thiophen-2-yl)-4H-pyran-4-one | CH...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208528(2-dibenzofuran-4-yl-6-morpholin-4-yl-pyran-4-one |...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50159678(3-Morpholin-4-yl-benzo[f]chromen-1-one | 3-morphol...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50132359(2-Morpholin-4-yl-6-phenyl-pyran-4-one | 2-morpholi...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208538(2-(4-methylnaphthalen-1-yl)-6-morpholino-4H-pyran-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208523(2-morpholino-6-(naphthalen-2-yl)-4H-pyran-4-one | ...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208530(2-(3-(benzyloxy)phenyl)-6-morpholino-4H-pyran-4-on...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208553(2-morpholino-6-(thiophen-3-yl)-4H-pyran-4-one | CH...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208529(4-morpholino-6-phenyl-2H-pyran-2-one | CHEMBL22140...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208517(2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one | C...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208537(CHEMBL222179 | benzyl 4-(6-morpholino-4-oxo-4H-pyr...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208508(6-(4-cyanophenyl)-2-morpholin-4-yl-4H-thiopyran-4-...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208513(2-morpholin-4-yl-6-thianthren-1-yl-4H-thiopyran-4-...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208524(2-morpholino-6-(naphthalen-1-yl)-4H-pyran-4-one | ...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50208534(3-(6-morpholino-4-oxo-4H-pyran-2-yl)benzaldehyde |...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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