Affinity DataIC50: 23nMAssay Description:Inhibition of KSP in KBV1 cells overexpressing PgpMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of KSP in KB31 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 123nMAssay Description:Inhibition of KSP in KBV1 cells overexpressing PgpMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of hERG expressed in CHO cells by cell voltage clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.59E+4nMAssay Description:Inhibition of hERG expressed in CHO cells by cell voltage clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.93E+4nMAssay Description:Inhibition of hERG expressed in CHO cells by cell voltage clamp assayMore data for this Ligand-Target Pair