Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50020031
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209698BDBM50209698(1-(3'-cyano-4-biphenylmethyl)-3-(2-hydroxy-1,1-dim...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209691BDBM50209691(1-(4'-fluoro-4-biphenylmethyl)-3-(2-hydroxy-1,1-di...)
Affinity DataKi:  96.6nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209692BDBM50209692(3-[1,1-di(hydroxymethyl)propyl]-1-(4'-methoxy-4-bi...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209693BDBM50209693(1-(4-biphenylmethyl)-3-(2-hydroxy-1,1-dimethylethy...)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209709BDBM50209709(1-(4'-fluoro-4-biphenylmethyl)-3-(1,1-di(hydroxyme...)
Affinity DataKi:  149nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209713BDBM50209713(3-[1,1-di(hydroxymethyl)propyl]-1-(2'-methoxy-4-bi...)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209699BDBM50209699(3-[1,1-di(acetyloxymethyl)propyl]-1-(4'-methoxy-4-...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209690BDBM50209690(1-(4-biphenylmethyl)-3-[1,1-di(hydroxymethyl)propy...)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209687BDBM50209687(1-(3'-cyano-4-biphenylmethyl)-3-[1-(4-methylbenzyl...)
Affinity DataKi:  186nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209711BDBM50209711(3-(2-hydroxy-1,1-dimethylethyl)-1-(4'-methoxy-4-bi...)
Affinity DataKi:  204nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209688BDBM50209688(3-[1,1-di(acetyloxymethyl)propyl]-1-(4'-fluoro-4-b...)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209689BDBM50209689(3-[1-(acetyloxymethyl)-1-methylethyl]-1-(2'-methox...)
Affinity DataKi:  215nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209717BDBM50209717(3-(2-hydroxy-1,1-dimethylethyl)-1-(2'-methoxy-4-bi...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209714BDBM50209714(3-[1-(acetyloxymethyl)-1-methylethyl]-1-(3'-cyano-...)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209707BDBM50209707(1-(4-biphenylmethyl)-3-isopropyl-1-{2-[1-(4-methyl...)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209715BDBM50209715(3-isopropyl-1-(4'-methoxy-4-biphenylmethyl)-1-{2-[...)
Affinity DataKi:  273nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209704BDBM50209704(1-(4'-fluoro-4-biphenylmethyl)-3-isopropyl-1-{2-[1...)
Affinity DataKi:  314nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209706BDBM50209706(3-[1,1-di(acetyloxymethyl)propyl]-1-(4-biphenylmet...)
Affinity DataKi:  388nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209700BDBM50209700(3-[1-(acetyloxymethyl)-1-methylethyl]-1-(4'-fluoro...)
Affinity DataKi:  421nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209705BDBM50209705(1-(2'-methoxy-4-biphenylmethyl)-3-[1-(4-methylbenz...)
Affinity DataKi:  425nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209702BDBM50209702(1-(3'-cyano-4-biphenylmethyl)-3-isopropyl-1-{2-[1-...)
Affinity DataKi:  509nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209694BDBM50209694(1-(4'-fluoro-4-biphenylmethyl)-3-[1-(4-methylbenzy...)
Affinity DataKi:  545nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209708BDBM50209708(3-[1-(acetyloxymethyl)-1-methylethyl]-1-(4'-methox...)
Affinity DataKi:  595nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209712BDBM50209712(1-(3'-cyano-4-biphenylmethyl)-3-[1,1-di(hydroxymet...)
Affinity DataKi:  769nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209695BDBM50209695(3-[1-(acetyloxymethyl)-1-methylethyl]-1-(4-bipheny...)
Affinity DataKi:  947nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209710BDBM50209710(3-[1,1-di(acetyloxymethyl)propyl]-1-(3'-cyano-4-bi...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209701BDBM50209701(3-[1,1-di(acetyloxymethyl)propyl]-1-(2'-methoxy-4-...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209697BDBM50209697(1-(4'-methoxy-4-biphenylmethyl)-3-[1-(4-methylbenz...)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209696BDBM50209696(1-(4-biphenylmethyl)-3-[1-(4-methylbenzyl)-4-piper...)
Affinity DataKi:  2.64E+3nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209686BDBM50209686(1-(4'-fluoro-4-biphenylmethyl)-1-(3-hydroxy-3-meth...)
Affinity DataKi:  5.86E+3nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209703BDBM50209703(1-(3-hydroxy-3-methyl-2-oxobutyl)-1-(2'-methoxy-4-...)
Affinity DataKi:  6.05E+3nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50209716BDBM50209716(1-(3'-cyano-4-biphenylmethyl)-1-(3-hydroxy-3-methy...)
Affinity DataKi:  6.38E+3nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed