Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50020167
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210886(1-(1-(3,4-dimethylbenzoyl)piperidin-4-yl)-1H-benzo...)
Affinity DataKi:  100nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210884(1-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)-1H...)
Affinity DataKi:  110nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210892(1-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)-4-...)
Affinity DataKi:  140nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210890(3-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)ben...)
Affinity DataKi:  170nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210901(1-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)-3-...)
Affinity DataKi:  180nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210899(1-(1-(4-amino-3-methoxybenzoyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  180nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210895(5-fluoro-1-(1-(3-methoxy-4-methylbenzoyl)piperidin...)
Affinity DataKi:  200nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210902(1-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)ind...)
Affinity DataKi:  240nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210898(3-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)ben...)
Affinity DataKi:  270nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210888(1-(1-(3-methoxybenzoyl)piperidin-4-yl)-1H-benzo[d]...)
Affinity DataKi:  300nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210905(1-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)-4,...)
Affinity DataKi:  330nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210904(5-chloro-1-(1-(3-methoxy-4-methylbenzoyl)piperidin...)
Affinity DataKi:  360nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210896(1-(1-(2-chloro-4-methoxypicolinoyl)piperidin-4-yl)...)
Affinity DataKi:  450nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210903(1-(1-(benzofuran-6-carbonyl)piperidin-4-yl)-1H-ben...)
Affinity DataKi:  500nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210894(5-chloro-1-(1-(3-methoxy-4-methylbenzoyl)piperidin...)
Affinity DataKi:  500nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210887(1-(1-(2,3-dimethylbenzoyl)piperidin-4-yl)-1H-benzo...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210897(1-(1-(benzo[d][1,3]dioxole-6-carbonyl)piperidin-4-...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210882(1-(1-(2-(trifluoromethyl)benzoyl)piperidin-4-yl)-1...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210889(1-(1-(4-tert-butylbenzoyl)piperidin-4-yl)-1H-benzo...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210885(1-(1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210891(1-(1-(4-(trifluoromethyl)benzoyl)piperidin-4-yl)-1...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210881(1-(1-(3-(trifluoromethyl)benzoyl)piperidin-4-yl)-1...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210900(1-(1-(2-fluorobenzoyl)piperidin-4-yl)-1H-benzo[d]i...)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210884(1-(1-(3-methoxy-4-methylbenzoyl)piperidin-4-yl)-1H...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 11betaHSD2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210906(1-(1-(furan-2-carbonyl)piperidin-4-yl)-1H-benzo[d]...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210893(1-(1-pivaloylpiperidin-4-yl)-1H-benzo[d]imidazol-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50210883(1-(1-(cyclohexanecarbonyl)piperidin-4-yl)-1H-benzo...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human 11-beta-HSD1 by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed