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Found 21 Enz. Inhib. hit(s) with all data for entry = 50020434
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM23823((2R)-2-amino-3-{[(4-methoxyphenyl)diphenylmethyl]s...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213730((R)-2-amino-3-(diphenyl(4-(trifluoromethyl)phenyl)...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213723((R)-methyl 2-amino-3-((4-methoxyphenyl)diphenylmet...)
Affinity DataIC50:  680nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM23772((2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanoi...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213727((R)-2-amino-3-(tritylthio)propanamide | CHEMBL2321...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM23812(CHEMBL232728 | S-Trityl-L-Cysteine (STLC) Analogue...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213733((R)-2-amino-3-((3,4-dimethoxyphenyl)diphenylmethyl...)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213734((R)-2-(((9H-fluoren-9-yl)methoxy)carbonyl)-3-(trit...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50109609((2R)-2-amino-3-mercaptopropanoic acid | (2R)-2-ami...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213731((R)-methyl 2-acetamido-3-((4-methoxyphenyl)dipheny...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM23808((2R)-2-acetamido-3-[(triphenylmethyl)sulfanyl]prop...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213729((R)-2-amino-3-(methylthio)propanoic acid | CHEMBL3...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213732((R)-2-amino-3-(2-aminoethylthio)propanoic acid | C...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM23809((2R)-2-[(triphenylmethyl)amino]-3-[(triphenylmethy...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213735((2R)-2-amino-3-[(carboxymethyl)sulfanyl]propanoic ...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM23811((2R)-2-{[(tert-butoxy)carbonyl]amino}-3-[(tripheny...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213728((R)-2-Amino-3-benzylsulfanyl-propionic acid | (R)-...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM23773((2R)-2-amino-3-[(diphenylmethyl)sulfanyl]propanoic...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213724((R)-2-Amino-3-(4-methoxy-benzylsulfanyl)-propionic...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213725((R)-2-amino-3-(tert-butylthio)propanoic acid | CHE...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Shizuoka

Curated by ChEMBL
LigandPNGBDBM50213726((R)-2-amino-3-[1-(9H-fluoren-9-yl)-meth-(E)-yliden...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibition of Eg5 assessed as inhibition ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed