Compile Data Set for Download or QSAR
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Found 17 Enz. Inhib. hit(s) with all data for entry = 50020494
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214523((R)-10-hydroxymethyl-6-methyl-5,6,6a,7-tetrahydro-...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214522((R)-2-methoxy-6,10-dimethyl-5,6,6a,7-tetrahydro-4H...)
Affinity DataKi:  21.5nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214523((R)-10-hydroxymethyl-6-methyl-5,6,6a,7-tetrahydro-...)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50036286((R)-(-)-10-methyl-11-hydroxyaporphine | (R)-6,10-d...)
Affinity DataKi:  216nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214522((R)-2-methoxy-6,10-dimethyl-5,6,6a,7-tetrahydro-4H...)
Affinity DataKi:  271nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214521((R)-10-hydroxymethyl-6-propyl-5,6,6a,7-tetrahydro-...)
Affinity DataKi:  375nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214520((R)-2-methoxy-10-methyl-6-propyl-5,6,6a,7-tetrahyd...)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]8-OH-DPAT from rat 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214520((R)-2-methoxy-10-methyl-6-propyl-5,6,6a,7-tetrahyd...)
Affinity DataKi:  1.35E+3nMAssay Description:Displacement of [3H]nemonapride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214523((R)-10-hydroxymethyl-6-methyl-5,6,6a,7-tetrahydro-...)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [3H]SCH23390 from rat dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214522((R)-2-methoxy-6,10-dimethyl-5,6,6a,7-tetrahydro-4H...)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [3H]SCH23390 from rat dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214521((R)-10-hydroxymethyl-6-propyl-5,6,6a,7-tetrahydro-...)
Affinity DataKi:  1.98E+3nMAssay Description:Displacement of [3H]SCH23390 from rat dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214520((R)-2-methoxy-10-methyl-6-propyl-5,6,6a,7-tetrahyd...)
Affinity DataKi:  2.79E+3nMAssay Description:Displacement of [3H]SCH23390 from rat dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214522((R)-2-methoxy-6,10-dimethyl-5,6,6a,7-tetrahydro-4H...)
Affinity DataKi:  3.76E+3nMAssay Description:Displacement of [3H]nemonapride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214521((R)-10-hydroxymethyl-6-propyl-5,6,6a,7-tetrahydro-...)
Affinity DataKi:  6.06E+3nMAssay Description:Displacement of [3H]nemonapride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50214523((R)-10-hydroxymethyl-6-methyl-5,6,6a,7-tetrahydro-...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of [3H]nemonapride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50036286((R)-(-)-10-methyl-11-hydroxyaporphine | (R)-6,10-d...)
Affinity DataKi:  9.65E+3nMAssay Description:Displacement of [3H]SCH23390 from rat dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50036286((R)-(-)-10-methyl-11-hydroxyaporphine | (R)-6,10-d...)
Affinity DataKi:  1.15E+4nMAssay Description:Displacement of [3H]nemonapride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed