Compile Data Set for Download or QSAR
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Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50020574
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215208(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-(2...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215203(1-(2,6-difluorobenzyl)-6-(4-chloro-2-methylbenzyl)...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215184((R)-1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-((...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215168(1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-(methy...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215223(1-(2,6-difluorobenzyl)-6-(4-(methylthio)benzyl)-3-...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215209(1-(2,6-difluorobenzyl)-3-(2-(methyl(2-(pyridin-2-y...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215165(1-(2,6-difluorobenzyl)-6-(4-(ethylthio)benzyl)-3-(...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215214(1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-(2-(me...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215218((R)-1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-((...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215204(1-(2,6-difluorobenzyl)-6-(4-ethylbenzyl)-3-(2-(met...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215193(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  25nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215179(1-(2,6-difluorobenzyl)-6-(4-(trifluoromethyl)benzy...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215211((R)-1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-((...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215190(1-(2,6-difluoro-benzyl)-6-(4-methyl-benzyl)-3-{2-[...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215221((R)-1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-(2...)
Affinity DataKi:  45nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215175((R)-1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-(2...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215177(1-(2-fluorobenzyl)-3-(2-(methyl(2-(pyridin-2-yl)et...)
Affinity DataKi:  80nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215217(1-(2,6-difluoro-benzyl)-6-(2-methyl-benzyl)-3-{2-[...)
Affinity DataKi:  85nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215173(1-(2,6-difluorobenzyl)-6-(4-methoxybenzyl)-3-(2-(m...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215191(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  160nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215188(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-(2...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215222(1-(2,6-difluorobenzyl)-6-(3,4-dichlorobenzyl)-3-(2...)
Affinity DataKi:  255nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215216(1-(2,6-difluorobenzyl)-6-(4-tert-butylbenzyl)-3-(2...)
Affinity DataKi:  300nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215170(1-benzyl-3-(2-(methyl(2-(pyridin-2-yl)ethyl)amino)...)
Affinity DataKi:  305nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215207(1-(cyclohexylmethyl)-3-(2-(methyl(2-(pyridin-2-yl)...)
Affinity DataKi:  380nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215174(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  490nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215180(6-(2-(1H-indol-3-yl)ethyl)-1-(2,6-difluorobenzyl)-...)
Affinity DataKi:  515nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215206(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  520nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215192(1-(2,6-difluoro-benzyl)-7-[4-imidazol-1-yl-benzyl]...)
Affinity DataKi:  540nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215219(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  600nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215182(1-(2,6-difluorobenzyl)-6-(4-(methylsulfonyl)benzyl...)
Affinity DataKi:  805nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215210(1-(2,6-difluorobenzyl)-6-(3-chlorobenzyl)-3-(2-(me...)
Affinity DataKi:  850nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215195(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  945nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215198(1-(2,6-difluoro-benzyl)-3-(3-methoxy-phenyl)-5,6,7...)
Affinity DataKi:  970nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215194(1-(2,6-difluoro-benzyl)-7-(2-methoxy-benzyl)-3-(3-...)
Affinity DataKi:  980nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215197(6-benzyl-1-(2,6-difluoro-benzyl)-3-{2-[methyl-(2-p...)
Affinity DataKi:  990nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215178(7-benzyl-1-(2,6-difluoro-benzyl)-3-(3-methoxy-phen...)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215215(1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-(((R)-...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215189((R)-1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-((...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215171(1-(2,6-difluorobenzyl)-6-(4-ethylbenzyl)-3-(2-(dim...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215172(1-(2,6-difluoro-benzyl)-7-[pyridin-4-yl-methyl]-3-...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215212(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215200(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-(2...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215220(1-(2,6-difluoro-benzyl)-7-[2-(1H-indol-3-yl)-ethyl...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215196((S)-1-(2,6-difluorobenzyl)-6-(4-chlorobenzyl)-3-((...)
Affinity DataKi:  2.41E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215213(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-(p...)
Affinity DataKi:  2.45E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215199(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  2.58E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215202(6-(2,4-dimethylbenzyl)-1-(2,6-difluorobenzyl)-3-((...)
Affinity DataKi:  2.59E+3nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215205(6-(3-methyl-benzo[b]thiophen-2-ylmethyl)-3-{2-[met...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50215176(1-(2,6-difluoro-benzyl)-7-[4-methylbenzyl]-3-(3-me...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I-His5,D-Tyr6]GnRH from human cloned GnRH receptor transfected in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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