Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50020761
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50200841(CHEMBL220360 | N-[(1S,2S)-3-(4-chlorophenyl)-2-(3-...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217220(N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)...)
Affinity DataIC50: 0.470nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217216(CHEMBL226642 | CHEMBL226591 | N-{(1S,2S)-2-(3-cyan...)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217216(CHEMBL226642 | CHEMBL226591 | N-{(1S,2S)-2-(3-cyan...)
Affinity DataIC50: 0.730nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217217(N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)...)
Affinity DataIC50: 0.770nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217213(N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217221(N-{(1S,2S)-2-(3-cyano-5-fluorophenyl)-3-[4-(2-fluo...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217222(N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217223(N-[(1S,2S)-2-(3-cyano-5-fluorophenyl)-3-(4-methoxy...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217218(N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)...)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217214(N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217224(N-{(1S,2S)-2-(3-cyanophenyl)-3-[4-(2-fluoroethoxy)...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217215(N-[(1S,2S)-2-(3-cyano-5-fluorophenyl)-3-[4-(fluoro...)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217216(CHEMBL226642 | CHEMBL226591 | N-{(1S,2S)-2-(3-cyan...)
Affinity DataIC50: 44nMAssay Description:Agonist activity at human CB2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed