Compile Data Set for Download or QSAR
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Report error Found 116 Enz. Inhib. hit(s) with all data for entry = 50020992
TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219717(CHEMBL246618 | N-(4-(3-bromophenyl)thiazol-2-yl)-4...)
Affinity DataEC50:  645nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219718(CHEMBL248426 | N-(2-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  7.90E+3nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219608(CHEMBL249062 | N-(4-(3-chloro-2-fluorophenyl)thiaz...)
Affinity DataEC50:  612nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219609(CHEMBL248434 | N-(3-(4-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219610(4-(1,2,4-triazin-3-ylamino)-N-(4-(2-fluoro-3-(trif...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219613(CHEMBL248218 | N-(4-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219614(CHEMBL249672 | N-(3-(4-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219612(CHEMBL249061 | N-(4-(2,3-difluorophenyl)thiazol-2-...)
Affinity DataEC50:  415nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219611(4-(1,3,5-triazin-2-ylamino)-N-(4-(2-fluoro-3-(trif...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219615(CHEMBL247650 | N-(4-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219616(CHEMBL249063 | N-(4-(3-bromo-2-fluorophenyl)thiazo...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219618(CHEMBL399768 | N-(1-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219623(CHEMBL247198 | N-(3-phenyl-1,2,4-thiadiazol-5-yl)-...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219622(CHEMBL429295 | N-(4-(2-fluoro-3-(trifluoromethoxy)...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219624(CHEMBL247641 | N-(4-(5-chloro-2-methoxyphenyl)thia...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219619(CHEMBL248428 | N-(3-(4-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219620(CHEMBL248026 | N-(5-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219630(CHEMBL247818 | N-(4-(2,4-dichlorophenyl)thiazol-2-...)
Affinity DataEC50:  510nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219629(CHEMBL245793 | N-(4-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219625(CHEMBL247606 | N-(4-(2-fluoro-3-(trifluoromethoxy)...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219627(CHEMBL399073 | N-(1-(3,4-dichlorophenyl)-1H-pyrazo...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219628(4-(2,6-dimethylpyrimidin-4-ylamino)-N-(4-(2-fluoro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219631(4-(pyrimidin-4-ylamino)-N-(4-(3-(trifluoromethoxy)...)
Affinity DataEC50:  284nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219633(4-(6-(azetidin-1-yl)pyrimidin-4-ylamino)-N-(4-(2-f...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219634(4-(6-(azetidin-1-yl)pyrimidin-4-ylamino)-N-(3-(4-f...)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219632(CHEMBL393268 | N-(4-(4-chloro-2-fluorophenyl)thiaz...)
Affinity DataEC50:  232nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219636(CHEMBL400559 | N-(4-(2-chlorophenyl)thiazol-2-yl)-...)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219635(4-(pyrimidin-4-ylamino)-N-(4-p-tolylthiazol-2-yl)b...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219637(4-(pyrimidin-4-ylamino)-N-(3-(3-(trifluoromethoxy)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219638(CHEMBL247822 | N-(4-(4-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219639(CHEMBL391597 | N-(4-(3,4-dichlorophenyl)thiazol-2-...)
Affinity DataEC50:  347nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219640(CHEMBL400869 | N-(3-(3,4-dichlorophenyl)-1,2,4-thi...)
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219642(CHEMBL399136 | N-(4-(4-chlorophenyl)thiazol-2-yl)-...)
Affinity DataEC50:  568nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219641(CHEMBL248047 | N-(3-(3,4-difluorophenyl)-1,2,4-thi...)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219621(4-(pyrimidin-4-ylamino)-N-(7-trifluoromethyl-4,5-d...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219649(CHEMBL397519 | N-(4-(2,6-dichloro-4-(trifluorometh...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219643(CHEMBL246847 | N-(4-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219644(CHEMBL248390 | N-(5-chloro-4-(4-fluoro-3-(trifluor...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219650(CHEMBL247041 | N-(4-(2-fluoro-3-isobutylphenyl)thi...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219648(CHEMBL248388 | N-(4-(4-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219647(4-(pyrimidin-4-ylamino)-N-(4-(2-(trifluoromethyl)p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219645(CHEMBL248042 | N-(4-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  84nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219646(CHEMBL247644 | N-(4-(2,3-difluoro-4-(trifluorometh...)
Affinity DataEC50:  87nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219654(CHEMBL440231 | N-(4-(2-fluoro-3-(trifluoromethyl)p...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219655(CHEMBL247461 | N-(4-(5-chloro-2-hydroxyphenyl)thia...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219656(CHEMBL247642 | N-(4-(3,4-difluorophenyl)thiazol-2-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219653(CHEMBL248055 | N-(3-(2-fluoro-3-(trifluoromethoxy)...)
Affinity DataEC50:  970nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219651(4-(pyrimidin-4-ylamino)-N-(4-(3-(trifluoromethyl)p...)
Affinity DataEC50:  418nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219662(4-(6-(ethylamino)pyrimidin-4-ylamino)-N-(4-(2-fluo...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThrombopoietin receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50219652(CHEMBL398549 | N-(4-(4-nitrophenyl)thiazol-2-yl)-4...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TPOr expressed in BaF3 cells by reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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