Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50003889
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440874BDBM50440874(CHEMBL398131)
Affinity DataEC50:  160nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477107BDBM50477107(CHEMBL410365)
Affinity DataEC50:  170nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440857BDBM50440857(CHEMBL392253)
Affinity DataEC50:  180nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477071BDBM50477071(CHEMBL266588)
Affinity DataEC50:  200nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440853BDBM50440853(CHEMBL236037)
Affinity DataEC50:  220nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440850BDBM50440850(CHEMBL238396)
Affinity DataEC50:  220nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440854BDBM50440854(CHEMBL236292)
Affinity DataEC50:  250nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440852BDBM50440852(CHEMBL414319)
Affinity DataEC50:  260nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440851BDBM50440851(CHEMBL267729)
Affinity DataEC50:  290nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477104BDBM50477104(CHEMBL235647)
Affinity DataEC50:  300nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440875BDBM50440875(CHEMBL236704)
Affinity DataEC50:  300nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477075BDBM50477075(CHEMBL410366)
Affinity DataEC50:  320nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440855BDBM50440855(CHEMBL236293)
Affinity DataEC50:  360nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440856BDBM50440856(CHEMBL398128)
Affinity DataEC50:  370nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440876BDBM50440876(CHEMBL396183)
Affinity DataEC50:  400nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440877BDBM50440877(CHEMBL397820)
Affinity DataEC50:  400nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477082BDBM50477082(CHEMBL396184)
Affinity DataEC50:  500nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477083BDBM50477083(CHEMBL439563)
Affinity DataEC50:  590nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477099BDBM50477099(CHEMBL237968)
Affinity DataEC50:  600nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477073BDBM50477073(CHEMBL278937)
Affinity DataEC50:  600nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477098BDBM50477098(CHEMBL236099)
Affinity DataEC50:  600nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477102BDBM50477102(CHEMBL237961)
Affinity DataEC50:  600nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440878BDBM50440878(CHEMBL438676)
Affinity DataEC50:  700nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477106BDBM50477106(CHEMBL236296)
Affinity DataEC50:  800nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477076BDBM50477076(CHEMBL236305)
Affinity DataEC50:  900nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477087BDBM50477087(CHEMBL238015)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477090BDBM50477090(CHEMBL235440)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477096BDBM50477096(CHEMBL266796)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477089BDBM50477089(CHEMBL393243)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477086BDBM50477086(CHEMBL236457)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477097BDBM50477097(CHEMBL236681)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477077BDBM50477077(CHEMBL266812)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477109BDBM50477109(CHEMBL398099)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477085BDBM50477085(CHEMBL237114)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477103BDBM50477103(CHEMBL397818)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477093BDBM50477093(CHEMBL237550)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477081BDBM50477081(CHEMBL438512)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477094BDBM50477094(CHEMBL398130)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477084BDBM50477084(CHEMBL266795)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477079BDBM50477079(CHEMBL410759)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477095BDBM50477095(CHEMBL237960)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477105BDBM50477105(CHEMBL237969)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477078BDBM50477078(CHEMBL396797)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477080BDBM50477080(CHEMBL238406)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477091BDBM50477091(CHEMBL398129)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477108BDBM50477108(CHEMBL236682)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477070BDBM50477070(CHEMBL238078)
Affinity DataEC50:  4.20E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477092BDBM50477092(CHEMBL236194)
Affinity DataEC50:  4.30E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477100BDBM50477100(CHEMBL236295)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProteinase-activated receptor 2(Human)
University of Queensland

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50477101BDBM50477101(CHEMBL395357)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at PAR2 expressed in human HT29 cells assessed as intracellular calcium releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
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